Target Details
| UniProt AC | P27448 |
|---|---|
| Gene Symbol | MARK3 |
| Protein Name | MAP/microtubule affinity-regulating kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02149 (KA1) PF00069 (Pkinase) PF00627 (UBA) |
Summary
- Multi-target molecules 170
- Clinical molecules 20
- Avg pChEMBL 6.74
Associated Diseases (1)
Active Molecules (170)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NFKMFNBKEOQNPZ
|
6.9 | Ki | 43 | — | |
PIQCTGMSNWUMAF
|
6.9 | Ki | 137 | Yes | |
QKFXSCNWJZKJSJ
|
6.9 | Ki | 7 | — | |
ALKJNCZNEOTEMP
|
6.9 | Kd | 55 | — | |
ZSZOBRBJIJWWHH
|
6.9 | IC50 | 4 | — | |
CFIBXVQLBVNOHW
|
6.8 | Ki | 64 | — | |
CLEGDJQQHUTCOW
|
6.8 | Ki | 43 | — | |
LUPCHAFIKZSOOK
|
6.8 | Ki | 15 | — | |
XFWUTMHVDGPWLH
|
6.8 | Ki | 75 | — | |
XPHWIERLJBFPFV
|
6.8 | Ki | 69 | — | |
YQKSNDNARJQAHP
|
6.8 | Ki | 12 | — | |
DBXGGXLBTWZXBB
|
6.7 | Ki | 39 | — | |
GDYZFFBMSBDTAA
|
6.7 | Ki | 60 | — | |
MZDKLVOWGIOKTN
|
6.7 | Ki | 80 | — | |
PSCJSWRVCKUMSL
|
6.7 | Ki | 35 | — | |
RKKIDHHGKNGTQI
|
6.7 | Ki | 28 | — | |
SBFPHSVZEXSHTL
|
6.7 | Ki | 62 | — | |
WINHZLLDWRZWRT
|
6.7 | Ki | 66 | — | |
YMIJUBCSOKSFRU
|
6.7 | Ki | 87 | — | |
KGPGFQWBCSZGEL
|
6.7 | Kd | 59 | Yes | |
JPOSFPUHBHRUAX
|
6.7 | IC50 | 40 | Yes | |
DYNHJHQFHQTFTP
|
6.7 | Kd | 38 | — | |
CKVWQORGCCEYHS
|
6.6 | Ki | 50 | — | |
JZTOUVBEZONDKA
|
6.6 | Ki | 80 | — | |
KKYPRNBBPBRJQX
|
6.6 | Ki | 40 | — | |
NJPWCTYVEJIQBM
|
6.6 | Ki | 72 | — | |
JOOXLOJCABQBSG
|
6.5 | Kd | 139 | — | |
AIQDZMUPVYDVLB
|
6.5 | Ki | 48 | — | |
AWDORCFLUJZUQS
|
6.5 | Ki | 22 | — | |
BQPLWJRDSDNGNE
|
6.5 | Ki | 16 | — | |
CHTMRWQLNNRRFJ
|
6.5 | Ki | 70 | — | |
FQYLJBVSYHZWLT
|
6.5 | Ki | 35 | Yes | |
MWKSRKSEWLRPBL
|
6.5 | Kd | 1075 | — | |
NKGLJTITEFZKAN
|
6.5 | Ki | 35 | — | |
WPHKIQPVPYJNAX
|
6.5 | Ki | 81 | — | |
YEHCNYAQEBQCCS
|
6.5 | Ki | 74 | — | |
IAYGCINLNONXHY
|
6.5 | Kd | 50 | — | |
UKBGBACORPRCGG
|
6.5 | IC50 | 17 | — | |
RYYNGWLOYLRZLK
|
6.4 | Kd | 45 | — | |
XKFTZKGMDDZMJI
|
6.4 | Kd | 64 | Yes | |
KOZFSFOOLUUIGY
|
6.4 | Kd | 88 | Yes | |
YFNWWNRZJGMDBR
|
6.4 | Kd | 35 | — | |
DFMCXVONDDGQIY
|
6.4 | Ki | 66 | — | |
GWJHMRBQEUHFOC
|
6.4 | Ki | 42 | — | |
IJNGXROUMFEKDB
|
6.4 | Ki | 39 | — | |
KWRXWPRFIUJQBP
|
6.4 | Ki | 25 | — | |
KXPWWMPXNUOYOH
|
6.4 | Ki | 24 | — | |
OADRBDVURCEKRP
|
6.4 | Ki | 44 | — | |
OUJZYQBEFNDJQN
|
6.4 | Ki | 71 | — | |
WAKGEHXTOOFEAE
|
6.4 | Ki | 27 | — |