Target Details
| UniProt AC | P27448 |
|---|---|
| Gene Symbol | MARK3 |
| Protein Name | MAP/microtubule affinity-regulating kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02149 (KA1) PF00069 (Pkinase) PF00627 (UBA) |
Summary
- Multi-target molecules 170
- Clinical molecules 20
- Avg pChEMBL 6.74
Associated Diseases (1)
Active Molecules (170)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.4 | Ki | 118 | — | |
HKSZLNNOFSGOKW
|
9.3 | IC50 | 408 | — | |
QNABDSWBQJKBHK
|
9.0 | IC50 | 45 | — | |
XLFNLJYGUOLEJS
|
8.9 | IC50 | 26 | — | |
HKSZLNNOFSGOKW
|
8.5 | Kd | 213 | — | |
OFIFLUFVENTCNZ
|
8.5 | IC50 | 11 | — | |
KRIUNPBAQZGFQA
|
8.4 | Ki | 76 | — | |
NGFGTMFVWSDFPS
|
8.3 | IC50 | 32 | — | |
OSVUGUHRKMMBSE
|
8.2 | Kd | 170 | — | |
UEFCSGDOOJJXTN
|
8.2 | IC50 | 46 | — | |
OWRXHGAFWZFFCW
|
8.2 | Ki | 113 | — | |
FLEAYYMORDPWAJ
|
8.1 | Ki | 90 | — | |
NLYZJYHBZFQGDP
|
8.0 | IC50 | 2 | — | |
UHEQNWGXIQUUOV
|
8.0 | IC50 | 2 | — | |
CLYMONPGUOMIQL
|
8.0 | Kd | 3 | — | |
QQWUGDVOUVUTOY
|
7.9 | Kd | 231 | Yes | |
NXSJMRCTGYTSTK
|
7.9 | Kd | 200 | — | |
LOZGENZISGZHOI
|
7.8 | IC50 | 2 | — | |
PBCZSGKMGDDXIJ
|
7.8 | Kd | 68 | Yes | |
RYYNGWLOYLRZLK
|
7.8 | Ki | 104 | — | |
OPSONJKOCBCHTM
|
7.7 | IC50 | 2 | — | |
VWVYILCFSYNJHF
|
7.7 | Ki | 49 | — | |
YOFJPZPGHXWQJB
|
7.7 | IC50 | 5 | — | |
BMGQWWVMWDBQGC
|
7.7 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
7.7 | Kd | 91 | Yes | |
MXHQJSWMMQETFE
|
7.6 | IC50 | 8 | — | |
APKZTNIHDKUHTG
|
7.6 | IC50 | 2 | — | |
ZUOYPKKUCQORTM
|
7.5 | IC50 | 2 | — | |
MVJMMLFMPWITEJ
|
7.5 | Ki | 110 | — | |
BSFNGHCTZDCQBF
|
7.4 | Ki | 93 | — | |
GCYXEGSPUDSZJY
|
7.4 | Ki | 82 | — | |
UIARLYUEJFELEN
|
7.3 | Kd | 289 | Yes | |
ADMFLILDQJSEIK
|
7.3 | Ki | 72 | — | |
FUMCKNCUEAQHCV
|
7.3 | Ki | 103 | — | |
RJZDECGDCKOHBV
|
7.3 | Ki | 70 | — | |
XKFTZKGMDDZMJI
|
7.3 | Ki | 56 | — | |
XYZNKCSDQRKAFR
|
7.3 | Ki | 53 | — | |
LRZYYIZFBXFSJB
|
7.2 | Ki | 69 | — | |
UMTWTCVTRDYHQQ
|
7.2 | Ki | 56 | — | |
ZGZVRPRSFXRGCF
|
7.2 | Ki | 76 | — | |
MHRZYVYAAMLZJC
|
7.1 | Ki | 4 | — | |
UDFDIIVNIYWXDM
|
7.1 | Ki | 74 | — | |
DASFSPDIWCMVRW
|
7.0 | Ki | 21 | — | |
PCQMERRARZKTPW
|
7.0 | Ki | 68 | — | |
PTVPBWWDGZSEAF
|
7.0 | Ki | 63 | — | |
ZWVZORIKUNOTCS
|
7.0 | Ki | 69 | — | |
AYCPARAPKDAOEN
|
7.0 | Kd | 73 | — | |
XUZMWHLSFXCVMG
|
7.0 | Kd | 24 | — | |
AILRADAXUVEEIR
|
6.9 | IC50 | 75 | — | |
FONINLXADYUZFI
|
6.9 | Ki | 25 | — |