Target Details
| UniProt AC | P27037 |
|---|---|
| Gene Symbol | ACVR2A |
| Protein Name | Activin receptor type-2A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF00069 (Pkinase) |
Summary
- Multi-target molecules 15
- Clinical molecules 3
- Avg pChEMBL 6.45
KEGG Pathways (4)
Active Molecules (15)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VAARYSWULJUGST
|
8.0 | Kd | 119 | Yes | |
MFAQYJIYDMLAIM
|
7.7 | Kd | 130 | Yes | |
CATARNNGBNYRJP
|
6.7 | IC50 | 2 | — | |
ZBNZXTGUTAYRHI
|
6.7 | Kd | 102 | Yes | |
PJNMAIKMKRLUIV
|
6.5 | IC50 | 3 | — | |
YYLKKYCXAOBSRM
|
6.5 | Kd | 191 | — | |
RGHVGCXGMWBBJX
|
6.2 | IC50 | 2 | — | |
QMOBMSIEJTZRFX
|
6.2 | IC50 | 2 | — | |
GYHQCQQLLQAFGA
|
6.1 | IC50 | 2 | — | |
PFTXFNSHFZLJNT
|
6.1 | IC50 | 17 | — | |
YSLKGORPFYLDEK
|
6.1 | IC50 | 2 | — | |
FBQRDQOHCIWKGC
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |