Target Details
| UniProt AC | P26639 |
|---|---|
| Gene Symbol | TARS1 |
| Protein Name | Threonine--tRNA ligase 1, cytoplasmic |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03129 (HGTP_anticodon) PF02824 (TGS) PF00587 (tRNA-synt_2b) PF07973 (tRNA_SAD) |
Summary
- Multi-target molecules 21
- Clinical molecules 0
- Avg pChEMBL 7.54
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (21)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MSFGWBJSNPMREF
|
8.9 | Ki | 2 | — | |
URBCTQBKEJDJNF
|
8.7 | Ki | 2 | — | |
SKSGONRDNZKNBF
|
8.5 | Ki | 2 | — | |
QIPHQMPGDDKWIL
|
8.5 | Ki | 2 | — | |
KUPGDBTUKULRSA
|
8.4 | Ki | 3 | — | |
TWJQKFNJORCUQW
|
8.3 | Ki | 2 | — | |
ZCCPLJOKGAACRT
|
8.3 | Kd | 599 | — | |
UZDQPUDWNCATGN
|
8.0 | Ki | 2 | — | |
UPVAPSGKXAAHBG
|
7.9 | Ki | 2 | — | |
UPVAPSGKXAAHBG
|
7.8 | IC50 | 2 | — | |
XIQXSKREZPNNJQ
|
7.5 | Ki | 2 | — | |
NUAFQODJAZYOPI
|
7.3 | Kd | 2 | — | |
MWKSRKSEWLRPBL
|
7.2 | Kd | 1075 | — | |
CTJLRNBGVURJQO
|
7.1 | Ki | 2 | — | |
DWJGNVFDIJMANO
|
7.0 | Ki | 2 | — | |
YUOYUTTYTCAEPF
|
6.9 | Kd | 2 | — | |
XJHNDUGHFDIXDU
|
6.9 | Kd | 2 | — | |
PZOVNOFAIPCMJX
|
6.4 | Ki | 2 | — | |
BTVLHQLQEFSMDM
|
6.3 | Ki | 2 | — | |
CKBTUCFDXHFPFY
|
6.2 | Ki | 2 | — | |
YAOLHMOKRGWWOB
|
6.0 | Ki | 2 | — |