Target Details
| UniProt AC | P26012 |
|---|---|
| Gene Symbol | ITGB8 |
| Protein Name | Integrin beta-8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF23106 (EGF_Teneurin) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 163
- Clinical molecules 0
- Avg pChEMBL 7.58
KEGG Pathways (11)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
Active Molecules (163)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LEBUVLVDRAIZDW
|
6.2 | IC50 | 5 | — | |
NOJLTMKHIVSHFR
|
6.2 | IC50 | 5 | — | |
STKPRFWUCQPKJQ
|
6.2 | IC50 | 3 | — | |
ADHOGOCWYMYMBV
|
6.1 | IC50 | 5 | — | |
APIKKGOIHMESQS
|
6.1 | IC50 | 5 | — | |
DCQCDEPHHWZADO
|
6.1 | IC50 | 4 | — | |
FZBGGWKHCWPGOF
|
6.1 | IC50 | 5 | — | |
KGVFBFPXRYIQHI
|
6.1 | IC50 | 5 | — | |
PBBRGHSUTCYOJM
|
6.1 | IC50 | 5 | — | |
BSLQJJPIELRITP
|
6.1 | IC50 | 7 | — | |
CCHDZAZXCIHJMH
|
6.0 | IC50 | 5 | — | |
IYLZCJGQHMLLPT
|
6.0 | IC50 | 5 | — | |
PLRHJUOUNRRNJH
|
6.0 | IC50 | 4 | — |