Target Details
| UniProt AC | P26012 |
|---|---|
| Gene Symbol | ITGB8 |
| Protein Name | Integrin beta-8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF23106 (EGF_Teneurin) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 163
- Clinical molecules 0
- Avg pChEMBL 7.58
KEGG Pathways (11)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
Active Molecules (163)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIIHYTXBJYTCBS
|
8.1 | IC50 | 4 | — | |
JOORNLXAAOZDNT
|
8.1 | IC50 | 3 | — | |
FVRPUSBGHNILEX
|
8.0 | IC50 | 3 | — | |
DRMIWPCMCBXOEN
|
8.0 | IC50 | 6 | — | |
JWYJAXVOVLDVAL
|
8.0 | IC50 | 6 | — | |
LXKNMILYYJXXKE
|
8.0 | IC50 | 6 | — | |
MPXAADAXXFWYMY
|
8.0 | IC50 | 7 | — | |
QESJLCKQPIPWOH
|
8.0 | IC50 | 4 | — | |
RZAGOFCCJINLJO
|
8.0 | IC50 | 6 | — | |
SFSRFYDTGQPIJA
|
8.0 | IC50 | 6 | — | |
ZDSIXCUNSXFSMQ
|
8.0 | IC50 | 6 | — | |
SGIGWAJIEAIDOA
|
8.0 | IC50 | 3 | — | |
IYESGKSMWJOJAX
|
7.9 | IC50 | 3 | — | |
CTIBSOFYGIAEHU
|
7.9 | IC50 | 3 | — | |
YTRFGUOSNFMZDW
|
7.9 | IC50 | 3 | — | |
IGUVQCZYMKVWFL
|
7.9 | IC50 | 3 | — | |
JLBKOTXUOFOXTK
|
7.8 | IC50 | 3 | — | |
KEVXOQVYLQXQLM
|
7.8 | IC50 | 3 | — | |
NIVBRIPUAQCFIE
|
7.8 | IC50 | 6 | — | |
OGWLKQKCWNAXLA
|
7.8 | IC50 | 5 | — | |
HGFOOLONGOBCMP
|
7.8 | IC50 | 6 | — | |
UTRLCJVXTOCKGU
|
7.7 | IC50 | 3 | — | |
DTTADTGUTFPRMD
|
7.7 | IC50 | 2 | — | |
HARYXLBGCPNWSN
|
7.7 | IC50 | 3 | — | |
AFSSMWIZDTYYKD
|
7.6 | IC50 | 3 | — | |
FLTIMXZSLYRKOV
|
7.6 | IC50 | 3 | — | |
FLTIMXZSLYRKOV
|
7.6 | IC50 | 6 | — | |
HKDUWRRLEDNORE
|
7.6 | IC50 | 6 | — | |
LWVBUNTVBHUROG
|
7.6 | IC50 | 3 | — | |
NTOCWOHJTCYCPV
|
7.6 | IC50 | 4 | — | |
WYADQJPQUJCCTC
|
7.6 | IC50 | 2 | — | |
DHKPZDWVBJIRBP
|
7.5 | IC50 | 6 | — | |
XJFNXAGFIMODFB
|
7.5 | IC50 | 3 | — | |
IJUIEQQTBTWZAD
|
7.5 | IC50 | 3 | — | |
LCFNLMPNEUINNK
|
7.5 | IC50 | 3 | — | |
JCYHCLYCEQLHFG
|
7.4 | IC50 | 3 | — | |
QJORAXWYSWNXGO
|
7.4 | IC50 | 3 | — | |
ZJLJEWROVSZOMN
|
7.4 | IC50 | 6 | — | |
GPLYJCNNOWRSTC
|
7.4 | IC50 | 4 | — | |
KXYAXQVLPNBUFO
|
7.4 | IC50 | 5 | — | |
CCJVTCXLUWYFKP
|
7.4 | IC50 | 3 | — | |
KEQKSJZXAMPQNA
|
7.4 | IC50 | 3 | — | |
FYTXCLMMODEFHA
|
7.3 | IC50 | 3 | — | |
YSRHKDWMDJOMGD
|
7.3 | IC50 | 3 | — | |
JPKURIUSIZMVHB
|
7.2 | IC50 | 3 | — | |
JOORNLXAAOZDNT
|
7.2 | IC50 | 3 | — | |
BXOSGYRJKCYDLH
|
7.2 | IC50 | 4 | — | |
YDNNKSZTMBYBMR
|
7.2 | IC50 | 3 | — | |
XWMGBLCMRLASDS
|
7.2 | IC50 | 8 | — | |
FUBVRQRCBDJFQQ
|
7.1 | IC50 | 6 | — |