Target Details
| UniProt AC | P26012 |
|---|---|
| Gene Symbol | ITGB8 |
| Protein Name | Integrin beta-8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23105 (EGF_integrin) PF23106 (EGF_Teneurin) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 163
- Clinical molecules 0
- Avg pChEMBL 7.58
KEGG Pathways (11)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
Active Molecules (163)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YLVNILLAZOYHHS
|
10.2 | IC50 | 6 | — | |
SHRSEUHJTZQLRO
|
9.7 | IC50 | 8 | — | |
YDHAGPCZRFQPOI
|
9.7 | IC50 | 6 | — | |
BQYBIJDRTDZCAJ
|
9.5 | IC50 | 8 | — | |
BWAUVRFZNDRMLY
|
9.5 | IC50 | 8 | — | |
GDEQKRGKHZOXGD
|
9.5 | IC50 | 8 | — | |
JXVVEFIKDDVLOS
|
9.5 | IC50 | 8 | — | |
QLBXWVBTUGYSGI
|
9.5 | IC50 | 8 | — | |
XRXSSPOFDFFALK
|
9.5 | IC50 | 8 | — | |
MFCABRSSOZYCRL
|
9.4 | IC50 | 8 | — | |
RTYLRDWEJUNBLU
|
9.4 | IC50 | 8 | — | |
YPAMHQMVIMQKOR
|
9.4 | IC50 | 8 | — | |
CJRDXSVCUSRJDR
|
9.3 | IC50 | 8 | — | |
QTBFGJFGHGTDRF
|
9.3 | IC50 | 8 | — | |
HIKDGFUZLZJZCB
|
9.2 | IC50 | 8 | — | |
OBOJFQICXTYCRY
|
9.2 | IC50 | 8 | — | |
BSNWAPOUYOPCPS
|
9.2 | IC50 | 6 | — | |
UCBYYQWMMNUSGH
|
9.2 | IC50 | 8 | — | |
PEFBVOAICYLSAF
|
9.0 | IC50 | 8 | — | |
ZAMKDPACDNUZPJ
|
9.0 | IC50 | 8 | — | |
CXHCNOMGODVIKB
|
8.9 | IC50 | 7 | — | |
WEVPEJCRRVAGCF
|
8.9 | IC50 | 3 | — | |
LDSSCYPSBICUEF
|
8.8 | IC50 | 3 | — | |
CVAFKDVZZYLXCZ
|
8.8 | IC50 | 6 | — | |
RZKTVFLXLRAPSQ
|
8.7 | IC50 | 3 | — | |
RRPRWSUXQMFYCJ
|
8.6 | IC50 | 3 | — | |
ZDUUJAZQZQAJEO
|
8.6 | IC50 | 6 | — | |
QZTBJCSOVXRYCX
|
8.5 | IC50 | 6 | — | |
HEVATADJCXEZNF
|
8.4 | IC50 | 3 | — | |
NLUXMQVEMDAZTJ
|
8.4 | IC50 | 6 | — | |
HFAIJFBXLXWVSM
|
8.4 | IC50 | 3 | — | |
GYEPIDGLKZAHSN
|
8.3 | IC50 | 3 | — | |
CJFKBQRLRONQOT
|
8.3 | IC50 | 7 | — | |
XQHLFZJLRICIOE
|
8.3 | IC50 | 6 | — | |
LPKVUBCTWTZOFS
|
8.2 | IC50 | 3 | — | |
BERIWRAMAHFVDY
|
8.2 | IC50 | 3 | — | |
ILKRHUYCJMCBRQ
|
8.2 | IC50 | 8 | — | |
RBJQMIIPTLTYFP
|
8.2 | IC50 | 8 | — | |
FUFDIYJXRSEIDD
|
8.2 | IC50 | 3 | — | |
NIHKLJCATASIRV
|
8.2 | IC50 | 6 | — | |
RZAGOFCCJINLJO
|
8.2 | IC50 | 6 | — | |
SRAAZWOKIPPIDS
|
8.2 | IC50 | 6 | — | |
YJXODXFHFQYURN
|
8.2 | IC50 | 6 | — | |
ZHKXSTJFXIMBBI
|
8.2 | IC50 | 6 | — | |
ZTDBHWGOQHAIQU
|
8.2 | IC50 | 3 | — | |
ZMXBIIQMSGOIRZ
|
8.2 | IC50 | 7 | — | |
AVTPXUYOKMVCFB
|
8.1 | IC50 | 3 | — | |
AVGZVNRRKZUYJJ
|
8.1 | IC50 | 6 | — | |
CJMISCRXEFTMEV
|
8.1 | IC50 | 6 | — | |
JXJGHJUDGYCRBL
|
8.1 | IC50 | 6 | — |