Target Details
| UniProt AC | P26010 |
|---|---|
| Gene Symbol | ITGB7 |
| Protein Name | Integrin beta-7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF08725 (Integrin_b_cyt) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 355
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Intestinal immune network for IgA production
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Transcriptional misregulation in cancer
Active Molecules (355)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IHTYXBYCVOIZGN
|
6.5 | IC50 | 3 | — | |
PQEXVAMKRQHKJU
|
6.5 | IC50 | 3 | — | |
QOPWOWOFTXTVMY
|
6.5 | IC50 | 3 | — | |
DBJXGLINUURUNI
|
6.5 | IC50 | 2 | — | |
JOYMVRZXGCGJQL
|
6.5 | IC50 | 2 | — | |
KFMZAEHOOJXIHH
|
6.5 | IC50 | 3 | — | |
RRHXZTGJYDPQIM
|
6.5 | IC50 | 3 | — | |
ZXQSUUGXCWMVCZ
|
6.5 | IC50 | 2 | — | |
FPRXGNGLIQZNBP
|
6.4 | IC50 | 2 | — | |
SQKRZWKSHPTTCU
|
6.4 | IC50 | 3 | — | |
XVFGXBXVSHPQNQ
|
6.4 | IC50 | 3 | — | |
RCBNMNQPHPCWME
|
6.4 | IC50 | 3 | — | |
ZIPHKIDWZBDOSS
|
6.4 | IC50 | 3 | — | |
FAQBNGGMUXLXSQ
|
6.4 | IC50 | 3 | — | |
ZCKOLWBSPNHKPQ
|
6.4 | IC50 | 2 | — | |
BNIJMUVCQMIEQC
|
6.4 | IC50 | 3 | — | |
NWAMIYLHUKLGAN
|
6.4 | IC50 | 3 | — | |
RZUNKWPPQAILPH
|
6.4 | IC50 | 3 | — | |
GSCDUHGSEPUEQF
|
6.4 | IC50 | 3 | — | |
KAUWYEHHOMTVRN
|
6.3 | IC50 | 3 | — | |
WPKLWLSFNMQEKC
|
6.3 | IC50 | 3 | — | |
BHTTYKCJLSWMIU
|
6.3 | IC50 | 3 | — | |
HPOGEWKAYYHIGE
|
6.3 | IC50 | 3 | — | |
ZYJZNWWXHXUROK
|
6.3 | IC50 | 3 | — | |
CCEPCRZUBCXDIG
|
6.3 | IC50 | 3 | — | |
GDLQGBLMGXDNRQ
|
6.3 | IC50 | 3 | — | |
OFQGKHJRPHPQFO
|
6.3 | IC50 | 2 | — | |
PJBWMOGSGAIFSM
|
6.3 | IC50 | 3 | — | |
APJVOWJJCXAZNW
|
6.3 | IC50 | 3 | — | |
ZXPQNPSQXMCMIJ
|
6.3 | IC50 | 3 | — | |
JOABXWLBYGYELJ
|
6.2 | IC50 | 3 | — | |
RCMILHNCCRVJJC
|
6.2 | IC50 | 3 | — | |
YNRFHLYLCWXFFX
|
6.2 | IC50 | 2 | — | |
UJHIRAKOONSSEL
|
6.2 | IC50 | 3 | — | |
PKPQFKVOUWIHGY
|
6.2 | IC50 | 3 | — | |
ACPZTVFLIFYRRX
|
6.2 | IC50 | 3 | — | |
NVVGCQABIHSJSQ
|
6.2 | IC50 | 6 | — | |
RVZYPCNWXCGBGD
|
6.2 | IC50 | 2 | — | |
CSMQOKNTHTXJFG
|
6.2 | IC50 | 3 | — | |
ZTQUXCXAZRNPHB
|
6.2 | IC50 | 2 | — | |
OYRUZFJXLJQJNA
|
6.2 | IC50 | 3 | — | |
PBIAFEAQIMQDNE
|
6.2 | IC50 | 3 | — | |
VNNBTSYVKBFTEF
|
6.2 | IC50 | 3 | — | |
CWYRXMARIDXJHG
|
6.2 | IC50 | 2 | — | |
PYLQHQVUGWACLR
|
6.1 | IC50 | 3 | — | |
TYGFNSSTUPFGIG
|
6.1 | IC50 | 3 | — | |
YTCSFWUXKXTEKH
|
6.1 | IC50 | 3 | — | |
CBPNUSPLCWQDTD
|
6.1 | IC50 | 3 | — | |
HHNBBKPRVOJRLK
|
6.1 | IC50 | 3 | — | |
HWDLYLCQKJBOBC
|
6.1 | IC50 | 2 | — |