Target Details
| UniProt AC | P26010 |
|---|---|
| Gene Symbol | ITGB7 |
| Protein Name | Integrin beta-7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF08725 (Integrin_b_cyt) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 355
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Intestinal immune network for IgA production
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Transcriptional misregulation in cancer
Active Molecules (355)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
APVDSPBBKYMHQH
|
6.8 | IC50 | 3 | — | |
XZFJCAFPBMJEOX
|
6.8 | IC50 | 3 | — | |
CGDRAVDJURFDMP
|
6.8 | IC50 | 3 | — | |
JHRWRZACLCUNPT
|
6.8 | IC50 | 3 | — | |
WCRJXUAYNQYKOD
|
6.8 | IC50 | 2 | — | |
IECKVUVUZIOYDW
|
6.8 | IC50 | 3 | — | |
BZEBVNQBGHZGIZ
|
6.8 | IC50 | 3 | — | |
CBFXJGDJKSJFLC
|
6.8 | IC50 | 2 | — | |
IGRGIQWZKAUHDT
|
6.8 | IC50 | 3 | — | |
NTFHSUUFBUDKFC
|
6.8 | IC50 | 3 | — | |
RBYPTCVDQLQTJV
|
6.8 | IC50 | 3 | — | |
MCUJFEQTPSDPLM
|
6.8 | IC50 | 3 | — | |
JVVBWVZYFIVRCL
|
6.8 | IC50 | 3 | — | |
BWSAPBQCDRMPGV
|
6.8 | IC50 | 2 | — | |
CJASQSIGTKSMFJ
|
6.8 | IC50 | 3 | — | |
DFGIRJIXSZXHRL
|
6.8 | IC50 | 3 | — | |
NVSCTWCNVXBLQP
|
6.8 | IC50 | 3 | — | |
WVTAFEUTNNWYQO
|
6.8 | IC50 | 3 | — | |
KIIRUEBNKLHWTL
|
6.7 | IC50 | 2 | — | |
YBKFCWABWAQJTN
|
6.7 | IC50 | 3 | — | |
CYOGWAISTADLSV
|
6.7 | IC50 | 3 | — | |
UERMUNMPBXMBHT
|
6.7 | IC50 | 3 | — | |
BZAIRWJDGMWPRS
|
6.7 | IC50 | 2 | — | |
RUVVTIYWVAZMKF
|
6.7 | IC50 | 3 | — | |
WQRWVWWUVJMCFW
|
6.7 | IC50 | 3 | — | |
XYXZMKHLXJARTF
|
6.7 | IC50 | 3 | — | |
SDRNIMLNYYTUKR
|
6.7 | IC50 | 3 | — | |
DAXUBPIJPVIZMQ
|
6.6 | IC50 | 3 | — | |
DSRYWCFQVDZVPR
|
6.6 | IC50 | 2 | — | |
KAPPMFUDCROIMR
|
6.6 | IC50 | 3 | — | |
DAEPHDSERDJBIQ
|
6.6 | IC50 | 3 | — | |
PMEZAVDXMBUKOU
|
6.6 | IC50 | 3 | — | |
RNWJDKPVADJMJR
|
6.6 | IC50 | 3 | — | |
PLNNIFRJWMGGGO
|
6.6 | IC50 | 3 | — | |
UAWIVFLVAQKETC
|
6.6 | IC50 | 3 | — | |
FWWQTACZOHEWIV
|
6.6 | IC50 | 2 | — | |
KNSNCKFGKKFIGH
|
6.6 | IC50 | 3 | — | |
IVZFOISXFATECM
|
6.6 | IC50 | 3 | — | |
RLDCURKHNWEZOG
|
6.6 | IC50 | 3 | — | |
IRWNJCIKJMZUEA
|
6.6 | IC50 | 2 | — | |
LPVTWENONSOHAO
|
6.6 | IC50 | 3 | — | |
IYGJJIDDHGARNB
|
6.6 | IC50 | 3 | — | |
AVOFTPGRAVVBLC
|
6.6 | IC50 | 3 | — | |
LXCVCICMQOFBDF
|
6.5 | IC50 | 2 | — | |
FXYDXLJEJBXFBD
|
6.5 | IC50 | 7 | — | |
JNMQDVKBQWASOW
|
6.5 | IC50 | 3 | — | |
GDSMXSYVAAVCRV
|
6.5 | IC50 | 3 | — | |
HJVXPUDBIZSBTO
|
6.5 | IC50 | 3 | — | |
JHRWRZACLCUNPT
|
6.5 | IC50 | 3 | — | |
TXTKZSBIOMEMHC
|
6.5 | IC50 | 3 | — |