Target Details
| UniProt AC | P26010 |
|---|---|
| Gene Symbol | ITGB7 |
| Protein Name | Integrin beta-7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF08725 (Integrin_b_cyt) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 355
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Intestinal immune network for IgA production
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Transcriptional misregulation in cancer
Active Molecules (355)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FOPAGNZNZJWJTG
|
7.1 | IC50 | 2 | — | |
OOKOWKFWBFLMMG
|
7.1 | IC50 | 2 | — | |
QFXPVNGZVLYJEY
|
7.1 | IC50 | 2 | — | |
SATRONDTGPPWOY
|
7.1 | IC50 | 3 | — | |
SFAOKQAQLNGQIZ
|
7.1 | IC50 | 3 | — | |
UKDPVOZZLJCIKT
|
7.1 | IC50 | 3 | — | |
MNQPNRJJCPTCFB
|
7.1 | IC50 | 2 | — | |
VNLCDFKUTJMNBN
|
7.1 | IC50 | 3 | — | |
LYHCGYLAKNFJSM
|
7.1 | IC50 | 3 | — | |
ACXGVBJSMSOQOF
|
7.1 | IC50 | 2 | — | |
CYRASILRFNUMJX
|
7.1 | IC50 | 3 | — | |
PXIBPFAADDDFDQ
|
7.1 | IC50 | 3 | — | |
WTUXQGQYRAGZCP
|
7.1 | IC50 | 3 | — | |
FJTPRDFOASDXPB
|
7.0 | IC50 | 3 | — | |
FOUDHXTZQKEKBC
|
7.0 | IC50 | 2 | — | |
HWPBTGQAYMMWRL
|
7.0 | IC50 | 2 | — | |
PLQYIPNBZHAKRA
|
7.0 | IC50 | 3 | — | |
CXISPJSWRIJOBE
|
7.0 | IC50 | 2 | — | |
HGEHCBNZQHVLJS
|
7.0 | IC50 | 3 | — | |
MIPYVVKAPSKISE
|
7.0 | IC50 | 2 | — | |
MNCLGSOOWQVRMZ
|
7.0 | IC50 | 2 | — | |
HXCSQLRXMBOJCE
|
7.0 | IC50 | 3 | — | |
BAILAXPMJUUBCX
|
7.0 | IC50 | 2 | — | |
LENTUXFIQXCWBP
|
7.0 | IC50 | 2 | — | |
LUQNTQZWQQXMQY
|
7.0 | IC50 | 3 | — | |
NSAOFDPAHXXLPO
|
7.0 | IC50 | 3 | — | |
DBTSBWISHCYWLW
|
7.0 | IC50 | 3 | — | |
VHYNCEYTMNADJU
|
7.0 | IC50 | 3 | — | |
SITGJFUZUFHSHU
|
7.0 | IC50 | 3 | — | |
LTQGACDEOSCTBA
|
7.0 | IC50 | 3 | — | |
UTLDJUNUIMQLSJ
|
7.0 | IC50 | 3 | — | |
GUIMDYNJLIADDB
|
7.0 | IC50 | 2 | — | |
LPTLKRBMBJHFHY
|
7.0 | IC50 | 3 | — | |
RNPDBUJJJTWLBJ
|
7.0 | IC50 | 2 | — | |
URESEGUVVXUPCQ
|
7.0 | IC50 | 2 | — | |
VEAVPXNJUXKCMP
|
6.9 | IC50 | 3 | — | |
CRFZTTKYQWZKDL
|
6.9 | IC50 | 2 | — | |
GPQMLRSUDYULCM
|
6.9 | IC50 | 2 | — | |
SFOPKWDSFYOUGN
|
6.9 | IC50 | 2 | — | |
KQFDKGNSBOLNCZ
|
6.9 | IC50 | 3 | — | |
UJSGTHFOHGFQMM
|
6.9 | IC50 | 3 | — | |
CEHJZAOMUIMHPN
|
6.9 | IC50 | 3 | — | |
IDUDYLQZZVVIFO
|
6.9 | IC50 | 3 | — | |
TXGRHCLDLARCJM
|
6.9 | IC50 | 3 | — | |
CAXSRPBPCGUCIY
|
6.8 | IC50 | 3 | — | |
SAYYIMRPRXVLIL
|
6.8 | IC50 | 3 | — | |
YUOMCSBLOMSMSI
|
6.8 | IC50 | 3 | — | |
DAEIMVCXNQVMSM
|
6.8 | IC50 | 3 | — | |
WRBJBMNRRSCTTO
|
6.8 | IC50 | 3 | — | |
YJBJPRUILPSVFT
|
6.8 | IC50 | 3 | — |