Target Details
| UniProt AC | P26010 |
|---|---|
| Gene Symbol | ITGB7 |
| Protein Name | Integrin beta-7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF08725 (Integrin_b_cyt) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 355
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Intestinal immune network for IgA production
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Transcriptional misregulation in cancer
Active Molecules (355)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FXYDXLJEJBXFBD
|
7.4 | IC50 | 6 | — | |
JGCUUCXMZKFRKP
|
7.4 | IC50 | 3 | — | |
LJSGBTCYWBYFTK
|
7.4 | IC50 | 3 | — | |
IBAZQIKVHCLTHH
|
7.4 | IC50 | 3 | — | |
REHPALZXYSKONM
|
7.4 | IC50 | 3 | — | |
DHPUSOIGQDLXGK
|
7.4 | IC50 | 2 | — | |
IAXOAOUFMTWSPG
|
7.4 | IC50 | 3 | — | |
JTVWJXUGGJTGDA
|
7.4 | IC50 | 4 | — | |
QRGLWLIXNHRUSY
|
7.4 | IC50 | 2 | — | |
SMZRAZWAVQZBEC
|
7.3 | IC50 | 3 | — | |
VVWWYYCPGHVEKY
|
7.3 | IC50 | 3 | — | |
BYRKTALPFLWGRH
|
7.3 | IC50 | 3 | — | |
DPTXHVXUQXOZLC
|
7.3 | IC50 | 3 | — | |
MCAIXYIMLUUTHW
|
7.3 | IC50 | 3 | — | |
NFMHJWOVOIOOTE
|
7.3 | IC50 | 3 | — | |
SLMLZSAUAQSGPC
|
7.3 | IC50 | 3 | — | |
KQRHUHXZMSKRIA
|
7.3 | IC50 | 2 | — | |
MOMXOJMYNNYSSO
|
7.3 | IC50 | 3 | — | |
DLBRECLYCZAQOF
|
7.3 | IC50 | 3 | — | |
LPPNDFOQUKQERO
|
7.3 | IC50 | 3 | — | |
WVPBLVXFXOYONK
|
7.3 | IC50 | 3 | — | |
LHDSVLWAOHWRLU
|
7.3 | IC50 | 3 | — | |
NOEWSRIYUKZVEG
|
7.3 | IC50 | 3 | — | |
OXXLQTUSOSKCPA
|
7.3 | IC50 | 2 | — | |
AEMBNJITTWJYBV
|
7.3 | IC50 | 3 | — | |
GNBZNYOXBLSXKD
|
7.3 | IC50 | 3 | — | |
KFNKHVGWGQDFPY
|
7.3 | IC50 | 3 | — | |
LDDBKVBDONLPAU
|
7.3 | IC50 | 3 | — | |
LTMQOAYQBDWTIQ
|
7.3 | IC50 | 3 | — | |
XFEBZCPSSQZCEA
|
7.3 | IC50 | 3 | — | |
LWMXBHHAGNVCLL
|
7.3 | IC50 | 3 | — | |
ROZGMDLHPFOJJF
|
7.3 | IC50 | 3 | — | |
GDOCTXXUSWKFKD
|
7.2 | IC50 | 3 | — | |
GSCXEBUWSNKNJK
|
7.2 | IC50 | 3 | — | |
HWTDZVDHOSKTML
|
7.2 | IC50 | 3 | — | |
XWJUDXXALXRTIE
|
7.2 | IC50 | 3 | — | |
HAFRWCGZNZNVIH
|
7.2 | IC50 | 3 | — | |
LCKQLWMWSSFPLR
|
7.2 | IC50 | 3 | — | |
WJGBWZYBCVVZMH
|
7.2 | IC50 | 2 | — | |
XMJDMDBLEIGQSK
|
7.2 | IC50 | 3 | — | |
YJMZWKYEAOOTFS
|
7.2 | IC50 | 3 | — | |
DLLGQRYZARKEBS
|
7.2 | IC50 | 3 | — | |
HJPINCWGHNTPPE
|
7.2 | IC50 | 2 | — | |
ROTDNRUETBXRKC
|
7.2 | IC50 | 2 | — | |
FNQSXZJGCVTEOX
|
7.2 | IC50 | 3 | — | |
SECAAPFNALWADD
|
7.2 | IC50 | 3 | — | |
KGMIDCRQGAMYTL
|
7.2 | IC50 | 2 | — | |
SQQCECFUGOZGKP
|
7.2 | IC50 | 3 | — | |
VDAVCTZCHJAJJR
|
7.2 | IC50 | 3 | — | |
ODFOVGIBIJCVKM
|
7.1 | IC50 | 3 | — |