Target Details
| UniProt AC | P26010 |
|---|---|
| Gene Symbol | ITGB7 |
| Protein Name | Integrin beta-7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF08725 (Integrin_b_cyt) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 355
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Intestinal immune network for IgA production
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Transcriptional misregulation in cancer
Active Molecules (355)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VFYLHJRNSIZWQQ
|
7.7 | IC50 | 3 | — | |
YZOVQSYKZPZDRM
|
7.7 | IC50 | 3 | — | |
IRVJBUBWERQASS
|
7.7 | IC50 | 3 | — | |
MXTOSAOISBOVCI
|
7.7 | IC50 | 3 | — | |
CMHZKJXTYSOXKN
|
7.7 | IC50 | 3 | — | |
CRLQMBSOODURJR
|
7.7 | IC50 | 3 | — | |
HOQJWEKHLQPATL
|
7.7 | IC50 | 2 | — | |
PGTKOGYRSWAQGX
|
7.7 | IC50 | 3 | — | |
VBHVOJJDISNENC
|
7.7 | IC50 | 3 | — | |
FPKILHQBPJHCHS
|
7.7 | IC50 | 3 | — | |
IJNZJGDRYIHSSV
|
7.7 | IC50 | 2 | — | |
OMKQSKNLFNSPII
|
7.7 | IC50 | 3 | — | |
VPIVICLWCZPBIT
|
7.7 | IC50 | 3 | — | |
YECQPPDRORMNRX
|
7.7 | IC50 | 3 | — | |
WGSFNDOOBOZLMA
|
7.7 | IC50 | 3 | — | |
FXYDXLJEJBXFBD
|
7.6 | IC50 | 6 | — | |
GJFNKTYJRCAGCV
|
7.6 | IC50 | 3 | — | |
RHXFXUSYPHIBOD
|
7.6 | IC50 | 3 | — | |
NVHYHKRZUDLBBQ
|
7.6 | IC50 | 3 | — | |
CUHMDYJWYPNQOZ
|
7.6 | IC50 | 2 | — | |
KSRNGDACGBIPKZ
|
7.6 | IC50 | 3 | — | |
WOZSUXNJFSSYJW
|
7.6 | IC50 | 3 | — | |
IGVOTDBZZXLCNQ
|
7.6 | IC50 | 3 | — | |
QSVHEGNXLMFWSO
|
7.6 | IC50 | 3 | — | |
YOVYUHGVQIKEOH
|
7.6 | IC50 | 2 | — | |
HISUKZFCUMSJFG
|
7.6 | IC50 | 3 | — | |
RTCKVCDARJCQAZ
|
7.6 | IC50 | 2 | — | |
DHLWZPYEINGBFR
|
7.6 | IC50 | 3 | — | |
AWGJFTQNOSRFEP
|
7.5 | IC50 | 3 | — | |
HUPHLMZTLJGDRG
|
7.5 | IC50 | 3 | — | |
JVMSOORAPUAHHJ
|
7.5 | IC50 | 2 | — | |
AQGOTKCWRZAUIP
|
7.5 | IC50 | 3 | — | |
BJHHYFPDNPOTHE
|
7.5 | IC50 | 4 | — | |
ULLBYKJYFPYRLS
|
7.5 | IC50 | 3 | — | |
VGUXHZDVUZBCSL
|
7.5 | IC50 | 2 | — | |
XUKXBXMAAGAYNG
|
7.5 | IC50 | 3 | — | |
WMXZKRJQWPXQIC
|
7.5 | IC50 | 2 | — | |
FRBLHLSRAGISCU
|
7.5 | IC50 | 2 | — | |
MEWSBKJAUCDJSK
|
7.5 | IC50 | 3 | — | |
PWLBENPPAZYTLF
|
7.5 | IC50 | 3 | — | |
ZGVJXSGTZGDJNP
|
7.5 | IC50 | 2 | — | |
LKNNQWMGOZFFKT
|
7.5 | IC50 | 3 | — | |
GZMUQYDHCNSVFL
|
7.4 | IC50 | 2 | — | |
KGDZUGSBEBVXKQ
|
7.4 | IC50 | 3 | — | |
RGCGVSJFGLIPEO
|
7.4 | IC50 | 3 | — | |
ZUYLZBWPGTXZOO
|
7.4 | IC50 | 3 | — | |
GIBVKJAUAVSEML
|
7.4 | IC50 | 2 | — | |
QVUGBFYAEPCUEO
|
7.4 | IC50 | 3 | — | |
VHCXDXCCKVQHGO
|
7.4 | IC50 | 2 | — | |
YGJLELVDLMNGTP
|
7.4 | IC50 | 3 | — |