Target Details
| UniProt AC | P26010 |
|---|---|
| Gene Symbol | ITGB7 |
| Protein Name | Integrin beta-7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF08725 (Integrin_b_cyt) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 355
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Intestinal immune network for IgA production
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Transcriptional misregulation in cancer
Active Molecules (355)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QODRKUNYZZPWLY
|
8.2 | IC50 | 3 | — | |
RROLERMMZPCBCQ
|
8.2 | IC50 | 2 | — | |
SSYLLNMYBQFPCH
|
8.2 | IC50 | 3 | — | |
DPLDYOSZVXSHEI
|
8.2 | IC50 | 3 | — | |
WKEYMRCHVPVMOY
|
8.2 | IC50 | 3 | — | |
DDXWRMMINAREGF
|
8.1 | IC50 | 3 | — | |
NKMZFGYUMYFYSM
|
8.1 | IC50 | 3 | — | |
RJALSTOENHOZQV
|
8.1 | IC50 | 3 | — | |
LBTMUQGNXSWGSG
|
8.1 | IC50 | 3 | — | |
MGAGDDCVRPUJAS
|
8.1 | IC50 | 3 | — | |
DMLHABDABMJTJN
|
8.0 | IC50 | 3 | — | |
IXDDZIVBYAEUTN
|
8.0 | IC50 | 3 | — | |
UYBXVMRNGPTDTI
|
8.0 | IC50 | 2 | — | |
AVPVBJWFJVXXIM
|
8.0 | IC50 | 3 | — | |
PALKXFSSVDMBNG
|
8.0 | IC50 | 3 | — | |
ZMKIAFJBCJTUFC
|
8.0 | IC50 | 3 | — | |
BKYBRLBEBOMPJQ
|
8.0 | IC50 | 3 | — | |
LGGGFIHRYYMBGJ
|
8.0 | IC50 | 3 | — | |
ADRBWUVQHKFVMS
|
7.9 | IC50 | 3 | — | |
AZIOXOMBBGKKBJ
|
7.9 | IC50 | 3 | — | |
KKZBAYODMNBMQJ
|
7.9 | IC50 | 3 | — | |
LAVKEKZSIBZMRJ
|
7.9 | IC50 | 3 | — | |
LBTMUQGNXSWGSG
|
7.9 | IC50 | 3 | — | |
NDJMYLPSHMDPKZ
|
7.9 | IC50 | 3 | — | |
OEJOIHNKFVHVEB
|
7.9 | IC50 | 3 | — | |
OZDFESSMPXWZSP
|
7.9 | IC50 | 3 | — | |
QSPRBGPZFIOHRF
|
7.9 | IC50 | 3 | — | |
ZNLSNWBYZFYQKK
|
7.9 | IC50 | 3 | — | |
GYNQANKDGGTNRK
|
7.9 | IC50 | 3 | — | |
OIIKLCMZNWWHNO
|
7.8 | IC50 | 3 | — | |
QYLJBVNSXNPXCO
|
7.8 | IC50 | 3 | — | |
CXSIVJHZBHTFAQ
|
7.8 | IC50 | 3 | — | |
HRZLYSAQTIAYDZ
|
7.8 | IC50 | 2 | — | |
NMSNKTZATNZHLY
|
7.8 | IC50 | 2 | — | |
POLDUUDTCKSSFP
|
7.8 | IC50 | 3 | — | |
YCYMAXCEGBEEOT
|
7.8 | IC50 | 3 | — | |
MWICRKHXHXGESF
|
7.8 | IC50 | 3 | — | |
YOCCTHZQHRBDCH
|
7.8 | IC50 | 3 | — | |
DAKQMEGZGHWYQY
|
7.8 | IC50 | 2 | — | |
AAQGLFLATBVJPM
|
7.8 | IC50 | 3 | — | |
MMIPQFQYOLUDRE
|
7.8 | IC50 | 3 | — | |
OGQYVSYKUNIBGC
|
7.8 | IC50 | 2 | — | |
FAXJBTWLKBIVML
|
7.8 | IC50 | 2 | — | |
FMKGFWRZZBCUCK
|
7.8 | IC50 | 2 | — | |
SCAJVSZKETYPPT
|
7.8 | IC50 | 3 | — | |
VVRIPMSPBSGFPZ
|
7.8 | IC50 | 3 | — | |
VVKWSNOGZODKEQ
|
7.7 | IC50 | 3 | — | |
GRCQDFIJVDYPTO
|
7.7 | IC50 | 2 | — | |
IILNCTZMDUGCHL
|
7.7 | IC50 | 3 | — | |
UCMTXIZUQCXQAO
|
7.7 | IC50 | 2 | — |