Target Details
| UniProt AC | P26010 |
|---|---|
| Gene Symbol | ITGB7 |
| Protein Name | Integrin beta-7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07974 (EGF_2) PF08725 (Integrin_b_cyt) PF00362 (Integrin_beta) PF17205 (PSI_integrin) |
Summary
- Multi-target molecules 355
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (13)
- Arrhythmogenic right ventricular cardiomyopathy
- Cell adhesion molecule (CAM) interaction
- Cytoskeleton in muscle cells
- Dilated cardiomyopathy
- ECM-receptor interaction
- Focal adhesion
- Human papillomavirus infection
- Hypertrophic cardiomyopathy
- Integrin signaling
- Intestinal immune network for IgA production
- PI3K-Akt signaling pathway
- Regulation of actin cytoskeleton
- Transcriptional misregulation in cancer
Active Molecules (355)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PDYIZJZZAUFVHP
|
9.6 | IC50 | 2 | — | |
UVGIBYJYUGXORP
|
9.5 | IC50 | 2 | — | |
NAKHAAQWKXWRKS
|
9.3 | IC50 | 2 | — | |
PWDOMNUZQXPHIM
|
9.2 | IC50 | 2 | — | |
DRSJLVGDSNWQBI
|
9.1 | IC50 | 4 | — | |
XRXLVYQWWZTNMN
|
9.1 | IC50 | 2 | — | |
XAENZKDUGMVTAX
|
9.0 | IC50 | 2 | — | |
RRBVGMXLNKTWFS
|
8.9 | IC50 | 2 | — | |
RIEDGQLYSUVDKT
|
8.8 | IC50 | 2 | — | |
QOXYYIKHVWXYGI
|
8.8 | IC50 | 2 | — | |
XDGSCLZNDKEXAE
|
8.7 | IC50 | 3 | — | |
BVCWBPBHALGRTA
|
8.7 | IC50 | 3 | — | |
LARLBZSTMWGXMK
|
8.7 | IC50 | 3 | — | |
SDQKXZWRNGVHOC
|
8.7 | IC50 | 3 | — | |
XYWVQRVWQOAUHV
|
8.7 | IC50 | 3 | — | |
YOUZAJBMSLTNRU
|
8.7 | IC50 | 3 | — | |
LPPNDFOQUKQERO
|
8.7 | IC50 | 3 | — | |
HZKMGPCRORUHHA
|
8.7 | IC50 | 2 | — | |
YPBWVSWHQCEYGY
|
8.7 | IC50 | 2 | — | |
UMWNDCFZURLHDU
|
8.6 | IC50 | 2 | — | |
UWDSAWYVWRSKPP
|
8.6 | IC50 | 3 | — | |
ZNCWUXZNXWDVRM
|
8.6 | IC50 | 2 | — | |
INVXYDDFZYTUMS
|
8.6 | IC50 | 2 | — | |
MGKZYWCSUHALDJ
|
8.6 | IC50 | 3 | — | |
CYCWDNHBPJXLCT
|
8.5 | IC50 | 3 | — | |
FUCBSFYEWUNIOP
|
8.5 | IC50 | 3 | — | |
OSQNFWWDIQJEHF
|
8.5 | IC50 | 3 | — | |
WYHTUAPAMDIATI
|
8.5 | IC50 | 3 | — | |
ZVKDMVSDTFKHRE
|
8.5 | IC50 | 3 | — | |
DXZXXIJEZVYUJW
|
8.5 | IC50 | 3 | — | |
XWZXOSXSUDVTSY
|
8.5 | IC50 | 3 | — | |
LDWAIULYHJTVQT
|
8.5 | IC50 | 3 | — | |
UTRBTIFHRKMFMU
|
8.5 | IC50 | 3 | — | |
AYPFNJVNXTYWGK
|
8.4 | IC50 | 3 | — | |
CIENDPDTDYSFMM
|
8.4 | IC50 | 3 | — | |
DVLBSXLUGBCBRC
|
8.4 | IC50 | 3 | — | |
NRCSJBQFSDHCEF
|
8.4 | IC50 | 2 | — | |
OCIRIHRFAHXBIT
|
8.4 | IC50 | 3 | — | |
JUBGULNNHUDWAO
|
8.4 | IC50 | 3 | — | |
PYDWJUFRRXINNH
|
8.3 | IC50 | 2 | — | |
ASYDYYRPDBLCFU
|
8.3 | IC50 | 3 | — | |
ASYDYYRPDBLCFU
|
8.3 | IC50 | 3 | — | |
PRUPKWNQAVQPOI
|
8.3 | IC50 | 3 | — | |
PSWUVNHTPHGXNB
|
8.3 | IC50 | 3 | — | |
WNKRETACHGJVKC
|
8.3 | IC50 | 3 | — | |
OPJBDVVJACDHPY
|
8.3 | IC50 | 3 | — | |
UZEJXLHLCJUOKN
|
8.3 | IC50 | 3 | — | |
GMZQXSJOGNIVAK
|
8.3 | IC50 | 3 | — | |
XYRKHQUYEVMHKJ
|
8.3 | IC50 | 3 | — | |
GMXTVNCMABOSEI
|
8.2 | IC50 | 3 | — |