Target Details
| UniProt AC | P25787 |
|---|---|
| Gene Symbol | PSMA2 |
| Protein Name | Proteasome subunit alpha type-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00227 (Proteasome) PF10584 (Proteasome_A_N) |
Summary
- Multi-target molecules 187
- Clinical molecules 0
- Avg pChEMBL 7.47
KEGG Pathways (8)
Active Molecules (187)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MLVUUPJRWINHGI
|
8.0 | IC50 | 19 | — | |
RXLPOAABTRQBFJ
|
8.0 | IC50 | 19 | — | |
KXNNVRZOLWDURQ
|
8.0 | IC50 | 19 | — | |
XNXFHORORFKFAC
|
8.0 | IC50 | 19 | — | |
GNHVWESRLVPKAE
|
8.0 | IC50 | 19 | — | |
HRIJMKFCVROBTA
|
7.9 | IC50 | 19 | — | |
PKEANJOUYSERAO
|
7.9 | IC50 | 38 | — | |
SOWWGFRAFDIXID
|
7.9 | IC50 | 20 | — | |
ZLCXYSYVRJMREV
|
7.9 | IC50 | 19 | — | |
RVKGLOJARNPYRU
|
7.8 | IC50 | 19 | — | |
MXAYKZJJDUDWDS
|
7.8 | IC50 | 22 | — | |
HDUYPFKWUPUIOZ
|
7.8 | IC50 | 19 | — | |
JEEJMGDWLRHOIC
|
7.8 | IC50 | 19 | — | |
MWKSRKSEWLRPBL
|
7.8 | Kd | 1075 | — | |
FHUUCFKFRIWULF
|
7.8 | IC50 | 19 | — | |
IINMCAOYFDMCLD
|
7.8 | IC50 | 19 | — | |
YKULOXYTLSPQGO
|
7.8 | IC50 | 19 | — | |
OGQMVFMKRZZEEH
|
7.7 | IC50 | 38 | — | |
ROOOPKPTTPSQLF
|
7.7 | IC50 | 19 | — | |
RSKYRPMOCHYBBE
|
7.7 | IC50 | 38 | — | |
XZXJGVCQHAWMAW
|
7.7 | IC50 | 19 | — | |
QKWHUQMFVKGCBD
|
7.7 | IC50 | 19 | — | |
YLKMLTBSIMGYTI
|
7.7 | IC50 | 19 | — | |
CFHYMTUYGRCJAV
|
7.7 | IC50 | 38 | — | |
FIHKCLKFORILIQ
|
7.7 | IC50 | 19 | — | |
WHPSHUGOCRYIEA
|
7.7 | IC50 | 20 | — | |
VMVVXXUNBWJIIZ
|
7.7 | IC50 | 38 | — | |
OWWIWRBLPZTZKF
|
7.7 | IC50 | 19 | — | |
CFFDAMKSIRGXAE
|
7.6 | IC50 | 19 | — | |
GAOQGHGKECEBBK
|
7.6 | IC50 | 38 | — | |
PFCGBSBLGKTTLF
|
7.6 | IC50 | 19 | — | |
SWZXEVABPLUDIO
|
7.6 | IC50 | 20 | — | |
DWBXJTGBTKJELX
|
7.6 | IC50 | 19 | — | |
QBPOBPNZSWZKFO
|
7.6 | IC50 | 19 | — | |
ATXBWTLLRQPRTF
|
7.6 | IC50 | 20 | — | |
QESQCTPAIQHKPZ
|
7.6 | IC50 | 19 | — | |
YVBOKFHQXPYEAC
|
7.6 | IC50 | 19 | — | |
MKGNEAHNDHHZJN
|
7.6 | IC50 | 19 | — | |
IJDYUMDIJFFMQQ
|
7.6 | IC50 | 19 | — | |
SAWUIOANDRGQBZ
|
7.6 | IC50 | 19 | — | |
XTGWWZCPEOEIIX
|
7.6 | IC50 | 19 | — | |
HSDWJRVETQTMBL
|
7.6 | IC50 | 19 | — | |
ODIWGDQSSAWSIL
|
7.5 | IC50 | 38 | — | |
SODXRIYSSYNQGD
|
7.5 | IC50 | 38 | — | |
UAKLEJZGAJPQOS
|
7.5 | IC50 | 19 | — | |
NBKCUYFBFZUFAE
|
7.5 | IC50 | 19 | — | |
VMNWBKJOXQEROK
|
7.5 | IC50 | 38 | — | |
XDCSOEDNLXDNQZ
|
7.5 | IC50 | 19 | — | |
WCTZLCQVQPYZIH
|
7.5 | IC50 | 19 | — | |
CRLANDXFFHDDAK
|
7.5 | IC50 | 20 | — |