Target Details
| UniProt AC | P25774 |
|---|---|
| Gene Symbol | CTSS |
| Protein Name | Cathepsin S |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 925
- Clinical molecules 1
- Avg pChEMBL 7.59
KEGG Pathways (5)
Active Molecules (925)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LEQCOSRDVNJGQU
|
7.8 | IC50 | 2 | — | |
RQFQNQBNKTWWPR
|
7.8 | IC50 | 3 | — | |
CXYMWYIUDRQGTR
|
7.8 | Ki | 2 | — | |
JBXZNIFMTVSEQN
|
7.8 | IC50 | 4 | — | |
SLXORIBUVHTOOX
|
7.8 | IC50 | 2 | — | |
XJZIQBQVGOEGFT
|
7.8 | Ki | 2 | — | |
YNWGZSVANLYSJR
|
7.8 | IC50 | 2 | — | |
BLJKFTVYZPTNBP
|
7.8 | Ki | 3 | — | |
ACGFKLACOBPYKQ
|
7.8 | IC50 | 4 | — | |
ACGFKLACOBPYKQ
|
7.8 | IC50 | 4 | — | |
AUHGCZBDMMKSIJ
|
7.8 | Ki | 2 | — | |
HRJIPNPMMDEUDH
|
7.8 | Ki | 3 | — | |
HSECIQLWCNQZCS
|
7.8 | Ki | 2 | — | |
KSKVGJIYFXPPFQ
|
7.8 | Ki | 2 | — | |
OZAFFYABJNEFEY
|
7.8 | Ki | 2 | — | |
QFJGHQXICGBKTL
|
7.8 | IC50 | 3 | — | |
SIIJWJNEODXHNY
|
7.8 | IC50 | 7 | — | |
SZYYBVWPURUFRR
|
7.8 | IC50 | 8 | — | |
UKNHAMBXKRGPNU
|
7.8 | Ki | 2 | — | |
VUNCDQVIHHNTRK
|
7.8 | Ki | 2 | — | |
XCVJGPONRKMMGU
|
7.8 | IC50 | 2 | — | |
ZGXKAZRUQQNMKC
|
7.8 | Ki | 3 | — | |
CRPZBEVSSSRFRT
|
7.8 | IC50 | 2 | — | |
GCWIICJLIHIUNY
|
7.8 | IC50 | 7 | — | |
GVIPJIBLWRMISS
|
7.8 | IC50 | 4 | — | |
IZZLPBCQUIYOGB
|
7.8 | IC50 | 4 | — | |
LWTHIEWNFZTHDQ
|
7.8 | IC50 | 4 | — | |
NJKWZQGOBIFPBG
|
7.8 | IC50 | 3 | — | |
ZBEYWPMZEAPAJQ
|
7.8 | IC50 | 2 | — | |
IKBUAFVMVGRIRN
|
7.8 | IC50 | 2 | — | |
CPDXLXNCBNKLMG
|
7.7 | IC50 | 4 | — | |
QCVFWWFGAKRNHR
|
7.7 | IC50 | 2 | — | |
RPFPLGIAONJHOM
|
7.7 | IC50 | 2 | — | |
AIBOMLIMFLTQOS
|
7.7 | IC50 | 3 | — | |
BJARUCXSUFPSCE
|
7.7 | IC50 | 2 | — | |
HBLWSGSCUSFXJE
|
7.7 | Ki | 3 | — | |
HMVXEHSUUNUEBL
|
7.7 | IC50 | 4 | — | |
QGJDTIUIQQOWOY
|
7.7 | Ki | 2 | — | |
IKTYGNJRDVXHJL
|
7.7 | IC50 | 2 | — | |
ADOJZMMSYUTJST
|
7.7 | IC50 | 2 | — | |
AJAZMOFONMJGNP
|
7.7 | IC50 | 3 | — | |
HFXHAUDVMVAJNA
|
7.7 | IC50 | 3 | — | |
KIBPLHFGSWCUTN
|
7.7 | IC50 | 2 | — | |
LTEDERVMQUPCSO
|
7.7 | IC50 | 3 | — | |
MECMHMVDUUQHDR
|
7.7 | Ki | 3 | — | |
MMOPUWHYSSYPDF
|
7.7 | IC50 | 2 | — | |
NMXQSPUYSZKXOQ
|
7.7 | IC50 | 2 | — | |
UHFLVCRUHSLCAK
|
7.7 | IC50 | 2 | — | |
VAIIZXKEFCDOFC
|
7.7 | IC50 | 2 | — | |
VSVZDJHBJJEDIL
|
7.7 | IC50 | 2 | — |