Target Details
UniProt ACP25774
Gene SymbolCTSS
Protein NameCathepsin S
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1)
Summary
  • Multi-target molecules 925
  • Clinical molecules 1
  • Avg pChEMBL 7.59
Top Co-occurrence Targets
Active Molecules (925)
InChIKey pChEMBL Type Targets Clinical
LTLYEAJONXGNFG 8.3 IC50 5
OZAJPIULESPARZ 8.3 Ki 2
BDSQVYWAMBOWIL 8.3 Ki 4
MNVJYJUEHVOPSA 8.3 IC50 2
YAGNDONYTVCOFN 8.3 IC50 3
FVZXHWVHTMNNBW 8.3 IC50 2
UAEAHQWORKLQQF 8.3 Ki 2
VJBNYTFCTIYDMG 8.3 IC50 3
FRXAKVHWABXMGZ 8.3 Ki 3
JGCPFQZBGQMKLG 8.3 IC50 2
RYZCDHLOJRGBKD 8.3 IC50 3
JUBANRFPTYBEFO 8.3 Ki 2
QTPYRNAKLBXKNP 8.3 IC50 3
SOFNUHHKAHJEAL 8.3 IC50 3
CJFRYKIQLJALCT 8.3 IC50 4
GLJZTHKUTGOBFU 8.3 Ki 4
GLMOVNGOIUEEJN 8.3 IC50 2
KPJQLFLWVFCIAV 8.3 IC50 2
KQXQLJBYHQUENE 8.2 Ki 3
AWEFNCACPBKWGG 8.2 Ki 3
MCKCVIDASJTQSU 8.2 Ki 3
BBMJJSLSNUWCEV 8.2 Ki 2
GMUXXTCOBZDVFS 8.2 Ki 4
TVUDUONIRJXXCP 8.2 Ki 4
DZZJCEAIGQTIHG 8.2 IC50 2
FJKPOCSUBVDARQ 8.2 IC50 3
GUBCDSPWYILVJH 8.2 IC50 4
IJVAYUWTLKHHKT 8.2 Ki 2
VMIIBGSXMXRAEG 8.2 IC50 2
YLLKTSVLFWTXPB 8.2 Ki 2
INALDMSSMJKKKP 8.2 IC50 2
LJJZYTHITLGKFY 8.2 IC50 2
OOVJOXGELNYKFE 8.2 IC50 3
BFHDYXSSAAUGPU 8.2 Ki 2
LTLYEAJONXGNFG 8.2 IC50 9
MTVNDTARQDTHDY 8.2 IC50 3
NNPAUJLJTFBVRA 8.2 Ki 2
SOHAERZROOTNSG 8.2 IC50 2
VHDAHAMWVNXMSP 8.2 IC50 7
YGYPGVCFJLTCGO 8.2 Ki 3
ZTDDKDQCLBTSDB 8.2 IC50 2
ZJMNNURDJNZLHH 8.1 Ki 3
BKBPVMYBRCWYHF 8.1 IC50 2
BKBPVMYBRCWYHF 8.1 IC50 2
CJDAPCDGESTEPR 8.1 Ki 4
FNEUKBQFZSGMQF 8.1 IC50 3
SYBYCMXFKUMMNW 8.1 IC50 4
UNICQUXWGGDNLF 8.1 Ki 4
UPGVOWXXAVOTAA 8.1 Ki 2
WDFFUHXXXVWAOH 8.1 Ki 2
2D structure