Target Details
| UniProt AC | P25774 |
|---|---|
| Gene Symbol | CTSS |
| Protein Name | Cathepsin S |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 925
- Clinical molecules 1
- Avg pChEMBL 7.59
KEGG Pathways (5)
Active Molecules (925)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SLQWQWLTTFJRHB
|
8.6 | IC50 | 2 | — | |
BNXDYZBRHZMVRA
|
8.6 | IC50 | 4 | — | |
UPWNNHRBMJWIBW
|
8.6 | IC50 | 3 | — | |
YOJBVDOLDVVFSO
|
8.6 | Ki | 2 | — | |
CRBJCNGWYFLJPW
|
8.6 | IC50 | 4 | — | |
GEOZVEILQGZHSF
|
8.6 | IC50 | 2 | — | |
KLKAVPREINBPNI
|
8.6 | IC50 | 2 | — | |
RHJLQMVZXQKJKB
|
8.6 | IC50 | 5 | — | |
YCPWFRMYSJKIIG
|
8.6 | IC50 | 4 | — | |
BUSQURRJWVUSJG
|
8.5 | IC50 | 2 | — | |
FBALKZAVEMIILY
|
8.5 | IC50 | 4 | — | |
JOBQWEVUTRQKOK
|
8.5 | IC50 | 3 | — | |
PYUCRBRSVPPZAU
|
8.5 | Ki | 2 | — | |
SVWMYRNQZSRCPR
|
8.5 | IC50 | 2 | — | |
WWVOULFEIOXZLF
|
8.5 | IC50 | 4 | — | |
FKLHWGFEHIHHIM
|
8.5 | IC50 | 2 | — | |
LGACDLUVLNDBOB
|
8.5 | IC50 | 4 | — | |
MGFZLEVVYSLEAX
|
8.5 | IC50 | 3 | — | |
PTUYLYPDSJMPGU
|
8.5 | IC50 | 2 | — | |
PUFJEFSFBMWBSG
|
8.5 | IC50 | 3 | — | |
QAGVIYYHBWIDBH
|
8.5 | IC50 | 3 | — | |
SHLWXCGNHANUPZ
|
8.5 | Ki | 2 | — | |
XJEBMYGPXQJVFF
|
8.5 | IC50 | 3 | — | |
YGPSKVNTXPFUTN
|
8.5 | IC50 | 3 | — | |
BBECUGKQKLZBOE
|
8.5 | Ki | 4 | — | |
JJFSLRIQURRAOH
|
8.5 | IC50 | 4 | — | |
CJBQZTNGRANTLJ
|
8.5 | IC50 | 2 | — | |
JRWQDVOHQWLANK
|
8.5 | Ki | 3 | — | |
DRNQQVHLNODFOO
|
8.5 | Ki | 2 | — | |
GZGBHAIADJLADQ
|
8.5 | IC50 | 4 | — | |
LWRWPGKGEKCHCZ
|
8.5 | Ki | 2 | — | |
LLYFTZCFPMXLKO
|
8.5 | IC50 | 2 | — | |
YOALWXUXVIVKNC
|
8.5 | IC50 | 2 | — | |
ZLUMYEPDTRVKBR
|
8.5 | IC50 | 2 | — | |
BWYBBMQLUKXECQ
|
8.4 | IC50 | 5 | — | |
ISMUQAIURWHJMU
|
8.4 | IC50 | 2 | — | |
KVMJONNVSMEASA
|
8.4 | Ki | 4 | — | |
OGRMAGULSQOTTD
|
8.4 | Ki | 4 | — | |
UDUSXNXRYOAZDW
|
8.4 | Ki | 2 | — | |
KWRWHECIURBTDP
|
8.4 | IC50 | 2 | — | |
DDBLZAUTWNNHGW
|
8.4 | IC50 | 2 | — | |
ZTZJEMIITUQFII
|
8.4 | Ki | 2 | — | |
QIZMDQBBKHFWJF
|
8.4 | Ki | 2 | — | |
CKWQDBSKPNIZBB
|
8.4 | IC50 | 3 | — | |
FQIORMPHDPHLKL
|
8.4 | IC50 | 2 | — | |
LQXJTYUJAKLJDS
|
8.4 | IC50 | 2 | — | |
TXNDJCXNKMIHRP
|
8.4 | Ki | 3 | — | |
ZTAFLDIJAATCDC
|
8.4 | Ki | 2 | — | |
VBPPNJCVXGAZDD
|
8.4 | Ki | 5 | — | |
CCFPTWLGKMFRNV
|
8.3 | IC50 | 2 | — |