Target Details
| UniProt AC | P25774 |
|---|---|
| Gene Symbol | CTSS |
| Protein Name | Cathepsin S |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 925
- Clinical molecules 1
- Avg pChEMBL 7.59
KEGG Pathways (5)
Active Molecules (925)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LBCGIKORTZAZTM
|
8.9 | IC50 | 3 | — | |
LZLJBBHMBQJUSF
|
8.9 | IC50 | 2 | — | |
QWIWJVVGLAKWBG
|
8.9 | IC50 | 4 | — | |
HCLPDRDQDGUFSD
|
8.8 | IC50 | 4 | — | |
JZLWWEAJMOECOO
|
8.8 | IC50 | 2 | — | |
FVTJPALETWZNEA
|
8.8 | IC50 | 2 | — | |
POPLFVJHDAWIDM
|
8.8 | IC50 | 3 | — | |
UTUSRLWZFBUDAM
|
8.8 | Ki | 4 | — | |
WTCANZGRFGLWSN
|
8.8 | IC50 | 3 | — | |
ZVFLOWMFPJEDHF
|
8.8 | IC50 | 2 | — | |
ALXQNHZWMOOFKL
|
8.8 | IC50 | 2 | — | |
CJTVJJOGOYUWJE
|
8.8 | IC50 | 2 | — | |
GUUHOTXBVVLLAX
|
8.8 | IC50 | 2 | — | |
XJKJCKLHFZWKFQ
|
8.8 | IC50 | 2 | — | |
YCJAZWGGWUWUMI
|
8.8 | IC50 | 2 | — | |
JPQIXMPQVCDFBY
|
8.8 | Ki | 5 | — | |
LCGRTAPRJZMTIT
|
8.7 | IC50 | 3 | — | |
PCJKSKCBOVMYIJ
|
8.7 | Ki | 4 | — | |
WHNDEIMPFCLXJS
|
8.7 | Ki | 4 | — | |
MLCSDXGMDJDAGE
|
8.7 | IC50 | 2 | — | |
BLXZSNSXPVRKAJ
|
8.7 | IC50 | 2 | — | |
NQJRWXSEROIEBL
|
8.7 | Ki | 2 | — | |
ROFMAUJRSYVSKK
|
8.7 | IC50 | 3 | — | |
ZGJILAJMKMDGOC
|
8.7 | IC50 | 4 | — | |
HJUPPNTXGDFNAO
|
8.7 | IC50 | 3 | — | |
KWAXBPZYRPIOSA
|
8.7 | Ki | 2 | — | |
NBEARLDWGIZSTM
|
8.7 | IC50 | 3 | — | |
NBJUMGLMSOHJOR
|
8.7 | IC50 | 2 | — | |
NLHKYJRHIGUIOQ
|
8.7 | IC50 | 2 | — | |
PFNHYFHJCWNICY
|
8.7 | IC50 | 2 | — | |
RHHVUDLUXPBHLT
|
8.7 | Ki | 3 | — | |
SNHOBOKULKSZIU
|
8.7 | Ki | 3 | — | |
YUICXLFAQWTQHG
|
8.7 | IC50 | 2 | — | |
AVAXSGXOQJUXHZ
|
8.7 | Ki | 2 | — | |
IVYNHONWIKUREB
|
8.7 | IC50 | 2 | — | |
VJIQEIGIVWRYOA
|
8.7 | IC50 | 2 | — | |
LMWXYUHYSBCVJI
|
8.7 | Ki | 3 | — | |
KODUWBVRDNFSES
|
8.6 | Ki | 2 | — | |
RTCASLUORPXCNR
|
8.6 | IC50 | 2 | — | |
UNCVRLMOEPDIDB
|
8.6 | Ki | 2 | — | |
VKQOQWWJCCFELL
|
8.6 | IC50 | 4 | — | |
XJKKWXRUCDAJHK
|
8.6 | IC50 | 4 | — | |
YYXKFKVZXGJJII
|
8.6 | IC50 | 2 | — | |
YFHSSOHMKVQRGY
|
8.6 | Ki | 2 | — | |
YJBKBVOKBCOKHA
|
8.6 | Ki | 2 | — | |
DGNCYEKXMJMVGO
|
8.6 | IC50 | 2 | — | |
AVUGRCORGNXBOQ
|
8.6 | IC50 | 4 | — | |
AVUGRCORGNXBOQ
|
8.6 | IC50 | 4 | — | |
GASCFELIQZXIAB
|
8.6 | IC50 | 3 | — | |
HBOZUMOKFHNMQI
|
8.6 | IC50 | 3 | — |