Target Details
| UniProt AC | P25774 |
|---|---|
| Gene Symbol | CTSS |
| Protein Name | Cathepsin S |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 925
- Clinical molecules 1
- Avg pChEMBL 7.59
KEGG Pathways (5)
Active Molecules (925)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OXGDHEYAOHZJLH
|
9.1 | IC50 | 2 | — | |
UXAHDVOIYHYCFE
|
9.1 | IC50 | 2 | — | |
WAWCVPQCGNEDNX
|
9.1 | IC50 | 4 | — | |
ADSUKSQQYWNBGE
|
9.1 | Ki | 2 | — | |
IJGGQKISOLMFMA
|
9.1 | IC50 | 2 | — | |
LHEWOPPODOUFHU
|
9.1 | IC50 | 4 | — | |
SKTUOKAQLMXSFD
|
9.1 | Ki | 2 | — | |
DSZHQXBJWZVALW
|
9.1 | IC50 | 2 | — | |
KQYFHIPAAHRARB
|
9.1 | Ki | 4 | — | |
PRXSBSULBZNTRC
|
9.1 | IC50 | 4 | — | |
XWMOCHXKDCBQPV
|
9.1 | Ki | 4 | — | |
YBSWDIITMXRJIB
|
9.1 | IC50 | 4 | — | |
DCDFVKDUIGKXRF
|
9.1 | Ki | 2 | — | |
GFHWMPSRNHRLNH
|
9.1 | IC50 | 2 | — | |
GJHYTSFTSOMLTG
|
9.1 | IC50 | 2 | — | |
HWNYTOPEHDSGOF
|
9.1 | IC50 | 3 | — | |
IWVHDBTWXSMDEF
|
9.0 | IC50 | 4 | — | |
WUXFAVQCMHVEHO
|
9.0 | IC50 | 2 | — | |
HEIHTFALJDNKRT
|
9.0 | IC50 | 4 | — | |
LKKLTPUNQSFPCU
|
9.0 | IC50 | 3 | — | |
AEACXIXTPAQTGN
|
9.0 | IC50 | 4 | — | |
AEWVXQSQQHUKLB
|
9.0 | IC50 | 2 | — | |
BTHLZKFLHOUZNZ
|
9.0 | Ki | 2 | — | |
GJSBZBUXDQKPBE
|
9.0 | IC50 | 2 | — | |
NSXOUETVXVPOFT
|
9.0 | IC50 | 4 | — | |
UOILZCHFKHELJR
|
9.0 | IC50 | 2 | — | |
XERMNVUWYPYRPN
|
9.0 | Ki | 3 | — | |
USPHVRZFPMWSPR
|
9.0 | IC50 | 4 | — | |
MEHDKDKCBBBTSM
|
9.0 | IC50 | 2 | — | |
XYMLZPAPBAMTAT
|
9.0 | IC50 | 2 | — | |
FMQLLJJKTLJHMC
|
9.0 | IC50 | 4 | — | |
KBOFMZZQYJBQLI
|
9.0 | IC50 | 2 | — | |
NSNODLMCUTYBRZ
|
9.0 | IC50 | 2 | — | |
SFTJBZSYFBMXOQ
|
9.0 | Ki | 2 | — | |
ULFKHVBAISSIOJ
|
9.0 | IC50 | 4 | — | |
VMSZYKRQEOLBRN
|
9.0 | IC50 | 2 | — | |
VMSZYKRQEOLBRN
|
9.0 | IC50 | 2 | — | |
YUMYYTORLYHUFW
|
9.0 | IC50 | 2 | — | |
BQWWAZOZDJROFE
|
8.9 | IC50 | 4 | — | |
IRSOCWQJNYLTDD
|
8.9 | IC50 | 2 | — | |
BVIAUHFJTQDKSF
|
8.9 | IC50 | 2 | — | |
OFNOZMJQFVWTHP
|
8.9 | IC50 | 4 | — | |
RIMTXKCDSVGCNW
|
8.9 | IC50 | 2 | — | |
YUMYYTORLYHUFW
|
8.9 | IC50 | 5 | — | |
BEEZUVIPTSBSGX
|
8.9 | IC50 | 2 | — | |
BHVRFNJEHAGAIV
|
8.9 | IC50 | 4 | — | |
FCADZVXWMPUWJQ
|
8.9 | IC50 | 2 | — | |
JUBWOHMBYIZWKV
|
8.9 | IC50 | 2 | — | |
DWNNWOUIBKMYHH
|
8.9 | Ki | 2 | — | |
JRUMBBNIAMXSAG
|
8.9 | IC50 | 3 | — |