Target Details
| UniProt AC | P25774 |
|---|---|
| Gene Symbol | CTSS |
| Protein Name | Cathepsin S |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 925
- Clinical molecules 1
- Avg pChEMBL 7.59
KEGG Pathways (5)
Active Molecules (925)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VZJRPBWJESTYLV
|
9.3 | IC50 | 4 | — | |
ZSTULDHUMOHIIR
|
9.3 | IC50 | 2 | — | |
UGAZRSHSXNNYTK
|
9.3 | Ki | 5 | — | |
XAPJBRQABYEJOX
|
9.3 | IC50 | 2 | — | |
ZNUMRCPRXWDFHV
|
9.3 | IC50 | 4 | — | |
HDQBKIWKLLGTGO
|
9.2 | IC50 | 4 | — | |
LBJZOWAHNPGWGP
|
9.2 | Ki | 3 | — | |
MZKPXTUNCMRSJY
|
9.2 | IC50 | 2 | — | |
RSEOJELKUSEFQD
|
9.2 | IC50 | 4 | — | |
UZEXNMTYYWVDSE
|
9.2 | IC50 | 4 | — | |
BFGMUSWYFUOFKU
|
9.2 | IC50 | 2 | — | |
GCILXAGICVRZQV
|
9.2 | IC50 | 4 | — | |
AHTSGKZDIBYODR
|
9.2 | Ki | 2 | — | |
BABQKRHMVVUNBI
|
9.2 | IC50 | 2 | — | |
KXNVRWXNNQCIBG
|
9.2 | IC50 | 2 | — | |
QSSXYXPPWDSHCS
|
9.2 | IC50 | 2 | — | |
QXLSWSCOFPRNEK
|
9.2 | IC50 | 4 | — | |
RHJLQMVZXQKJKB
|
9.2 | IC50 | 5 | — | |
VZSXPUDQSLKVIR
|
9.2 | Ki | 4 | — | |
WDFRBUOXDFQBFN
|
9.2 | IC50 | 2 | — | |
YYVYNDITYXLIBI
|
9.2 | IC50 | 4 | — | |
ZEFHIBBPLAGQMT
|
9.2 | IC50 | 2 | — | |
FFZKUHOGZGQBST
|
9.2 | IC50 | 2 | — | |
HBSWEZXYFZOCOH
|
9.2 | IC50 | 4 | — | |
KIDPFKMKRUSRRX
|
9.2 | IC50 | 4 | — | |
NILSEPPHIUAUFQ
|
9.2 | IC50 | 4 | — | |
LNFFLKXYCXMVTE
|
9.2 | IC50 | 4 | — | |
MCYQKGNJBOSMKC
|
9.2 | IC50 | 4 | — | |
HSRHZZRELKYVLU
|
9.2 | IC50 | 2 | — | |
YRDWNESAGCXMTG
|
9.2 | IC50 | 4 | — | |
ZIUAFVCBRREUMS
|
9.2 | IC50 | 2 | — | |
ACTMEZFPDCIVQO
|
9.2 | IC50 | 2 | — | |
GAJNSRVTRDPQFO
|
9.2 | IC50 | 2 | — | |
OPOAWRFREKKVNV
|
9.2 | IC50 | 2 | — | |
HOYOWCXIOGAMFB
|
9.2 | IC50 | 2 | — | |
IPZZWADNXFGPHL
|
9.2 | IC50 | 2 | — | |
KCWJNSONIBRYMQ
|
9.2 | IC50 | 2 | — | |
OQVJUAAFCYLUII
|
9.2 | IC50 | 4 | — | |
QTUJLNUNFRGPFA
|
9.2 | IC50 | 2 | — | |
TWOOZSOQPIWDLA
|
9.2 | IC50 | 3 | — | |
VLROHFCAQABUTJ
|
9.2 | IC50 | 3 | — | |
LQPSYXJJLUINTM
|
9.1 | IC50 | 2 | — | |
PUMWIMQYYHNBAM
|
9.1 | IC50 | 4 | — | |
ZBRHHBWBGUXOAL
|
9.1 | IC50 | 4 | — | |
ZPOFUECDFORWNJ
|
9.1 | IC50 | 2 | — | |
WGVGLTXVMMTGKM
|
9.1 | IC50 | 3 | — | |
FTQLFUOHNOGLNP
|
9.1 | Ki | 4 | — | |
GGWWZSKHPHUDIG
|
9.1 | IC50 | 4 | — | |
NBCJOXDJIAVNOB
|
9.1 | IC50 | 2 | — | |
ORVBPDVWWASNIP
|
9.1 | IC50 | 2 | — |