Target Details
| UniProt AC | P25774 |
|---|---|
| Gene Symbol | CTSS |
| Protein Name | Cathepsin S |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 925
- Clinical molecules 1
- Avg pChEMBL 7.59
KEGG Pathways (5)
Active Molecules (925)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XXCXONRLKKHITM
|
10.6 | Ki | 3 | — | |
JRHFOWQWUVMCHX
|
9.9 | Ki | 5 | — | |
UEZMKFGTDYYCKL
|
9.9 | IC50 | 3 | — | |
AUPZRAAKTGPDLC
|
9.8 | Ki | 4 | — | |
CLOALCKDNZPWBO
|
9.8 | Ki | 4 | — | |
MWBPTVRPPPPZPG
|
9.8 | Ki | 4 | — | |
LRGPAVMYPWWORG
|
9.8 | Ki | 4 | — | |
LHJKRUYOLRIDGD
|
9.8 | Ki | 4 | — | |
ARWSHTCIMVGBCQ
|
9.7 | Ki | 4 | — | |
BXOVKTMPLLKCSP
|
9.7 | IC50 | 3 | — | |
HRRZJMMKIKNUDN
|
9.7 | IC50 | 3 | — | |
JESRGSWARNNMLP
|
9.7 | Ki | 4 | — | |
SCCNQBNFEHNRCO
|
9.7 | Ki | 4 | — | |
SEBANXBXZIIACF
|
9.7 | IC50 | 3 | — | |
YZBDFADJOLGKFN
|
9.6 | IC50 | 3 | — | |
QVDJMLQSYRSZKC
|
9.6 | Ki | 6 | Yes | |
UZMSYDMWVBDKEM
|
9.5 | IC50 | 4 | — | |
AXVMAPSVAWPASZ
|
9.5 | Ki | 3 | — | |
GLDNCRGNTMYXND
|
9.5 | IC50 | 3 | — | |
LJPQZPJJLKMWAU
|
9.5 | IC50 | 2 | — | |
SQIHYRIDUCIHLT
|
9.5 | IC50 | 2 | — | |
KFTMZNIURYIOKI
|
9.5 | Ki | 4 | — | |
PFCKPTDNLNORNL
|
9.5 | IC50 | 2 | — | |
GZBOGFDHJAMENH
|
9.5 | Ki | 4 | — | |
PYZOXRXOZRPQAH
|
9.5 | IC50 | 4 | — | |
JEBQNHANRCYVLC
|
9.5 | IC50 | 4 | — | |
DEKMUSVVANPFAA
|
9.4 | IC50 | 4 | — | |
CGGQUYWUIFSOCV
|
9.4 | IC50 | 2 | — | |
NWBGYSJMEUHJPR
|
9.4 | IC50 | 2 | — | |
TYRHHAXPGPFWOM
|
9.4 | IC50 | 2 | — | |
CDUNEFIKZYZKAG
|
9.4 | IC50 | 2 | — | |
SLSHNBKPDGBYGO
|
9.4 | IC50 | 3 | — | |
XAHPKDQGKQJQGR
|
9.4 | IC50 | 3 | — | |
VZTRAYHUTKYOCB
|
9.4 | IC50 | 4 | — | |
FLCQJGNOUMHLTG
|
9.4 | IC50 | 2 | — | |
NRLBGKWSOSYHJM
|
9.4 | IC50 | 4 | — | |
NWFXZBFOOLIBAC
|
9.3 | IC50 | 2 | — | |
ZZPFZJXGGZUTHR
|
9.3 | IC50 | 4 | — | |
AJGQRLLAZUYHKK
|
9.3 | IC50 | 2 | — | |
BLQYPJAWNZQHRK
|
9.3 | IC50 | 2 | — | |
KZCODYXMOKIMLT
|
9.3 | IC50 | 3 | — | |
NOTSCKFHTQJLMM
|
9.3 | IC50 | 3 | — | |
PJOCENBBWQXQGY
|
9.3 | Ki | 3 | — | |
UWIUSTCLSVVZSO
|
9.3 | IC50 | 3 | — | |
XSAIUGYZCYGLEW
|
9.3 | IC50 | 2 | — | |
YJZKURYVZRISEA
|
9.3 | IC50 | 2 | — | |
CAQLLDUOKIHSBN
|
9.3 | IC50 | 3 | — | |
FTJHEEIVOBBMMC
|
9.3 | Ki | 5 | — | |
YGOOSESWCCPOHN
|
9.3 | IC50 | 4 | — | |
UHNROXZSASTRFP
|
9.3 | IC50 | 4 | — |