Target Details
| UniProt AC | P25440 |
|---|---|
| Gene Symbol | BRD2 |
| Protein Name | Bromodomain-containing protein 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 699
- Clinical molecules 0
- Avg pChEMBL 7.25
Active Molecules (699)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RJPKAAVNTLYQAC
|
7.2 | IC50 | 3 | — | |
STSKCRDOTKSTPF
|
7.2 | IC50 | 3 | — | |
YNMSRPUOAQPYLV
|
7.2 | IC50 | 3 | — | |
PXLJQXYHONWMKB
|
7.2 | IC50 | 3 | — | |
SMYPWBHABVYAJK
|
7.2 | IC50 | 3 | — | |
UZPOOTYPBOTHKT
|
7.2 | IC50 | 3 | — | |
BHZGECKOYMLRSO
|
7.2 | IC50 | 3 | — | |
FUOUPXXFTDVPGM
|
7.2 | IC50 | 3 | — | |
KLKMODXQLGKDKQ
|
7.2 | Ki | 3 | — | |
PDCBJZVPIGAEBL
|
7.2 | IC50 | 4 | — | |
QSLHPKXGYOTUHN
|
7.2 | IC50 | 3 | — | |
SKTNIECRSURWAZ
|
7.2 | IC50 | 3 | — | |
WPRFMKAORZZEIZ
|
7.2 | IC50 | 3 | — | |
SDLMPYCGZKLARA
|
7.2 | IC50 | 4 | — | |
SUIIIOQGACLJMI
|
7.2 | IC50 | 3 | — | |
UVCPBOQPPSLUPY
|
7.2 | IC50 | 3 | — | |
PIKWYDHWUKSWAQ
|
7.2 | Kd | 4 | — | |
DAXLHHYYMDQRCH
|
7.2 | IC50 | 3 | — | |
IEEQBCSZMPIUGM
|
7.2 | IC50 | 3 | — | |
JFLRJPGRSNHGAL
|
7.2 | IC50 | 3 | — | |
LWGUCDPMTIPABX
|
7.2 | IC50 | 4 | — | |
RKSYSKOBHCWHKB
|
7.2 | IC50 | 3 | — | |
SJSCJYHUBPKPNG
|
7.2 | IC50 | 3 | — | |
WCNXRFKEDHKCLC
|
7.2 | IC50 | 3 | — | |
XBQGLWPUGBREQS
|
7.2 | IC50 | 4 | — | |
XNRZMTWJFLFRMR
|
7.2 | IC50 | 3 | — | |
FAWSUKOIROHXAP
|
7.2 | IC50 | 5 | — | |
GQXFGAMRIGUNFT
|
7.2 | IC50 | 4 | — | |
PXLJQXYHONWMKB
|
7.2 | IC50 | 3 | — | |
GKJNYZBASPYBEP
|
7.2 | IC50 | 3 | — | |
KOWPYSXWLGSRKS
|
7.2 | IC50 | 2 | — | |
LCXHXIMNUYTCEI
|
7.2 | IC50 | 3 | — | |
LFNLJQQQSRYUHQ
|
7.2 | IC50 | 3 | — | |
PQYXGDZAWKQEEM
|
7.2 | IC50 | 3 | — | |
DDIGBXFXYQBMSG
|
7.1 | IC50 | 3 | — | |
FFHFKSXIZXKTRE
|
7.1 | IC50 | 3 | — | |
FMJBUHAFPYWEKA
|
7.1 | IC50 | 3 | — | |
OYMMHSBUFOLNEY
|
7.1 | IC50 | 3 | — | |
UFFMFBORABJCTA
|
7.1 | Ki | 3 | — | |
VVRZMYLMDPVHTL
|
7.1 | Ki | 3 | — | |
WQRKDXUDKMFKPL
|
7.1 | IC50 | 4 | — | |
PASBWKAEFYVJHG
|
7.1 | IC50 | 3 | — | |
SJACAKNFJFXOJF
|
7.1 | IC50 | 3 | — | |
HKECFOZBEGKIAX
|
7.1 | IC50 | 3 | — | |
IVXYIGADMWHQDD
|
7.1 | IC50 | 4 | — | |
MSZSAGAHXQKHRZ
|
7.1 | IC50 | 3 | — | |
OZPNRBXVIUPSDJ
|
7.1 | Kd | 4 | — | |
QGIHDISRDFTWAD
|
7.1 | IC50 | 3 | — | |
UYRUHHLEYUGTMC
|
7.1 | IC50 | 3 | — | |
DNVXATUJJDPFDM
|
7.1 | Kd | 4 | — |