Target Details
| UniProt AC | P25440 |
|---|---|
| Gene Symbol | BRD2 |
| Protein Name | Bromodomain-containing protein 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 699
- Clinical molecules 0
- Avg pChEMBL 7.25
Active Molecules (699)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VVSCZWKYDATSNC
|
7.3 | IC50 | 3 | — | |
WODOTYIRVRGFSJ
|
7.3 | IC50 | 3 | — | |
BSZDTJJAUVZTBS
|
7.3 | IC50 | 3 | — | |
GQXFGAMRIGUNFT
|
7.3 | IC50 | 4 | — | |
UZPOOTYPBOTHKT
|
7.3 | IC50 | 3 | — | |
XRQOPEVIGOZEJD
|
7.3 | IC50 | 3 | — | |
ZBKQSWPCHUEZBL
|
7.3 | IC50 | 3 | — | |
BRAMSTZRKUJRKS
|
7.3 | IC50 | 4 | — | |
BRAMSTZRKUJRKS
|
7.3 | IC50 | 3 | — | |
CPWCZLPJMXCWDY
|
7.3 | IC50 | 3 | — | |
FLASGTNYMYVYKJ
|
7.3 | IC50 | 3 | — | |
MDRXOFSNECSECW
|
7.3 | Ki | 3 | — | |
MMMRGZLSUKMQOD
|
7.3 | IC50 | 4 | — | |
UQMYMWRETIHSGQ
|
7.3 | IC50 | 3 | — | |
UYBRROMMFMPJAN
|
7.3 | Kd | 8 | — | |
VAXZYGLGDOWBGT
|
7.3 | IC50 | 3 | — | |
ABSZIZKRSYKAPX
|
7.3 | IC50 | 4 | — | |
AEOQRVQQPVQSRQ
|
7.3 | IC50 | 3 | — | |
GAVLMQAIIHDXBG
|
7.3 | IC50 | 2 | — | |
KOWPYSXWLGSRKS
|
7.3 | IC50 | 3 | — | |
NCEJUIVQBWZGMA
|
7.3 | IC50 | 3 | — | |
NYYPYDLZLGCKOU
|
7.3 | IC50 | 4 | — | |
SJACAKNFJFXOJF
|
7.3 | IC50 | 2 | — | |
TUWDLUFFAHHNEF
|
7.3 | Kd | 3 | — | |
TUWDLUFFAHHNEF
|
7.3 | Kd | 3 | — | |
WQEGQSRMXSLEON
|
7.3 | IC50 | 3 | — | |
YTYPEASDFWXHLK
|
7.3 | IC50 | 3 | — | |
ZQFOFTHJENGQKG
|
7.3 | IC50 | 3 | — | |
DNVXATUJJDPFDM
|
7.3 | IC50 | 17 | — | |
MVAYDDZVYGANLI
|
7.3 | IC50 | 3 | — | |
NVRXYLMWFKVLJI
|
7.3 | IC50 | 3 | — | |
UHWGSUFICDUCKV
|
7.3 | IC50 | 3 | — | |
ZOVYOHAZPIKVOR
|
7.3 | IC50 | 4 | — | |
DFHREBKXJWXHKG
|
7.3 | Kd | 2 | — | |
HIZNONHBBUUYFX
|
7.3 | IC50 | 4 | — | |
IMXDUOIANVGJIA
|
7.3 | IC50 | 3 | — | |
QXTHZAMLLIIJHM
|
7.3 | IC50 | 3 | — | |
AURWSPRKUDZZIW
|
7.2 | IC50 | 3 | — | |
FZFLGRAVZYFGBB
|
7.2 | Kd | 4 | — | |
GVCFSBGCJBRHFS
|
7.2 | IC50 | 4 | — | |
MVAYDDZVYGANLI
|
7.2 | IC50 | 3 | — | |
VVPPHMRXPGDFBQ
|
7.2 | IC50 | 3 | — | |
ZNGYYGUCWRDEAS
|
7.2 | IC50 | 3 | — | |
KOYGJJMRJVPCNS
|
7.2 | IC50 | 3 | — | |
UBXNLHDUJFHNDS
|
7.2 | IC50 | 3 | — | |
BNWMHKNZCUUJMF
|
7.2 | IC50 | 3 | — | |
CQPGVZBZRUVJJZ
|
7.2 | IC50 | 3 | — | |
FUXOAMWDPVPAFQ
|
7.2 | IC50 | 3 | — | |
MZKIOOQWOZDDMX
|
7.2 | IC50 | 3 | — | |
OENGVXVRDHPNME
|
7.2 | IC50 | 3 | — |