Target Details
| UniProt AC | P25440 |
|---|---|
| Gene Symbol | BRD2 |
| Protein Name | Bromodomain-containing protein 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 699
- Clinical molecules 0
- Avg pChEMBL 7.25
Active Molecules (699)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YJEIXSZAEKFWTM
|
7.4 | IC50 | 3 | — | |
JNYUGWPUYNNZOZ
|
7.4 | Kd | 3 | — | |
JVTTVFOTQZIFEV
|
7.4 | IC50 | 3 | — | |
PYJQEIWIODYCRH
|
7.4 | IC50 | 3 | — | |
VUWJZAUOMZSUEU
|
7.4 | IC50 | 3 | — | |
AMRTUWDHDGIYSC
|
7.4 | IC50 | 3 | — | |
GKJNYZBASPYBEP
|
7.4 | IC50 | 3 | — | |
IMBCMESWDHPIDA
|
7.4 | IC50 | 3 | — | |
JKTAXQJDSRMHSS
|
7.4 | IC50 | 3 | — | |
PKHUSSXCMLLVRI
|
7.4 | IC50 | 3 | — | |
VLVRBRZAFGCGJV
|
7.4 | IC50 | 3 | — | |
BUFWGONUWXTMGP
|
7.4 | IC50 | 3 | — | |
BUFWGONUWXTMGP
|
7.4 | IC50 | 3 | — | |
FRDVUWTYVBTBSE
|
7.4 | IC50 | 3 | — | |
HQEUJXGKBKBFIW
|
7.4 | IC50 | 3 | — | |
HSMCUAMXZNQLSQ
|
7.4 | IC50 | 3 | — | |
OFFYQYIVOWBZLD
|
7.4 | IC50 | 3 | — | |
QLRYSHYUZMZZPY
|
7.4 | IC50 | 3 | — | |
WEHPZXXDBNJUIG
|
7.4 | IC50 | 3 | — | |
WKDIHLGAKPCUJV
|
7.4 | IC50 | 3 | — | |
WUFYDWKEOKQEEP
|
7.4 | IC50 | 3 | — | |
IUUGMLRGSKSQJD
|
7.4 | IC50 | 3 | — | |
NEUUJGUKAZAFHZ
|
7.4 | IC50 | 3 | — | |
RIDHDDTVNQHKEQ
|
7.4 | IC50 | 3 | — | |
SRFOIWNXIILSNJ
|
7.4 | IC50 | 4 | — | |
VFDAORCFAAAXRV
|
7.4 | IC50 | 3 | — | |
XZYFNQNYLMTZIS
|
7.4 | IC50 | 3 | — | |
ZSBDKRBBDNFMHY
|
7.4 | Ki | 3 | — | |
ZZJIAOWVSKZQGQ
|
7.4 | IC50 | 3 | — | |
AWVPNUWHMBPXOU
|
7.4 | Kd | 8 | — | |
GLMGIYSAZNFOHX
|
7.4 | IC50 | 3 | — | |
IOHXSSTYGFWMFM
|
7.4 | IC50 | 3 | — | |
IVJMCRKXIOARPS
|
7.4 | IC50 | 3 | — | |
RWRYTMPXTGYISG
|
7.4 | IC50 | 3 | — | |
WQBRHFBWJUCVRR
|
7.4 | IC50 | 3 | — | |
QWMJOPLEXJAKPN
|
7.4 | IC50 | 3 | — | |
BWMCWOZPWHUTGN
|
7.3 | IC50 | 3 | — | |
DVICYEUYFBDIJO
|
7.3 | IC50 | 3 | — | |
NJQDQDHZAAGIQX
|
7.3 | IC50 | 3 | — | |
HDHIHYNEQCFQNL
|
7.3 | IC50 | 3 | — | |
KLPMURBFDSDZSU
|
7.3 | IC50 | 3 | — | |
OQBRSKHYDQIBJE
|
7.3 | IC50 | 3 | — | |
GAFAVXVVQUWUQX
|
7.3 | IC50 | 3 | — | |
GZEDEKFDZMUCGJ
|
7.3 | IC50 | 4 | — | |
JADOFDPLHYUWBU
|
7.3 | IC50 | 3 | — | |
OYDMPDMTZYTSSQ
|
7.3 | IC50 | 3 | — | |
FTHLNVOKHACXIU
|
7.3 | IC50 | 3 | — | |
KBQLHGZSZFKGCG
|
7.3 | IC50 | 3 | — | |
SNDFCVARRAHINB
|
7.3 | IC50 | 3 | — | |
SNXGAWWAXJMADO
|
7.3 | IC50 | 3 | — |