Target Details
| UniProt AC | P25440 |
|---|---|
| Gene Symbol | BRD2 |
| Protein Name | Bromodomain-containing protein 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 699
- Clinical molecules 0
- Avg pChEMBL 7.25
Active Molecules (699)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LVOINJWONMUWBO
|
7.5 | IC50 | 2 | — | |
MLMDKPAWBXFXNA
|
7.5 | IC50 | 3 | — | |
MYTABVRHXGACGI
|
7.5 | IC50 | 4 | — | |
SVEGTFMYOXJKMY
|
7.5 | IC50 | 3 | — | |
XNRZMTWJFLFRMR
|
7.5 | IC50 | 4 | — | |
CBNDXTMVECMPGV
|
7.5 | IC50 | 4 | — | |
KKQGFFSHWVTNMA
|
7.5 | IC50 | 3 | — | |
MGLUYQBSWDKFIR
|
7.5 | IC50 | 3 | — | |
OGJPTYDTRCDEJC
|
7.5 | IC50 | 3 | — | |
SNBMTDIABWCKJS
|
7.5 | IC50 | 2 | — | |
SWZWWWDWBVBZDV
|
7.5 | IC50 | 3 | — | |
YJEIXSZAEKFWTM
|
7.5 | IC50 | 3 | — | |
YXHZTVCEXBXXJR
|
7.5 | IC50 | 3 | — | |
FFMRDJNJHCWRIX
|
7.5 | IC50 | 3 | — | |
KDRSWORUPZEOGX
|
7.5 | IC50 | 3 | — | |
WGJDGQSSFHDLIX
|
7.5 | IC50 | 3 | — | |
XZYFNQNYLMTZIS
|
7.5 | IC50 | 3 | — | |
YSAPPGXSSQEHTA
|
7.5 | IC50 | 3 | — | |
LMYKZDUQLVXDIX
|
7.5 | IC50 | 3 | — | |
NEOVBISHUWMCQM
|
7.5 | IC50 | 3 | — | |
PXTNXIAHIKBHPF
|
7.5 | IC50 | 3 | — | |
RYGFKPUPLGKCHY
|
7.5 | IC50 | 3 | — | |
SJSCJYHUBPKPNG
|
7.5 | IC50 | 3 | — | |
TWYGARCNNFAUNW
|
7.5 | IC50 | 3 | — | |
ZBKQIKDKLUJFMK
|
7.5 | Ki | 3 | — | |
ZFJHDWKVFUWKQS
|
7.5 | IC50 | 3 | — | |
DGXUFGAFFVEFEU
|
7.4 | IC50 | 3 | — | |
FBYKSRDDFYPNNO
|
7.4 | IC50 | 3 | — | |
FRDRCUWLVRNFIJ
|
7.4 | IC50 | 3 | — | |
LMQMHIFIMOPETK
|
7.4 | IC50 | 3 | — | |
MGLUYQBSWDKFIR
|
7.4 | IC50 | 3 | — | |
WIFZFGUMQICZOO
|
7.4 | IC50 | 3 | — | |
XYJCDALAOYQCIB
|
7.4 | IC50 | 2 | — | |
ZDMWQHIIHYYGIB
|
7.4 | IC50 | 3 | — | |
ZJTYXGWJNWESQV
|
7.4 | Kd | 3 | — | |
ZUEZEQZVGBUYFN
|
7.4 | IC50 | 3 | — | |
FFHFKSXIZXKTRE
|
7.4 | IC50 | 3 | — | |
KKLVVGZXBWABFO
|
7.4 | IC50 | 3 | — | |
LMCSAEHKLPKZOO
|
7.4 | IC50 | 3 | — | |
LZYVFLZEQAANSW
|
7.4 | IC50 | 3 | — | |
UCJMBWXOKLINTN
|
7.4 | IC50 | 4 | — | |
WYUJMOVTXOPUEX
|
7.4 | IC50 | 4 | — | |
ZKVURPUQVABYSC
|
7.4 | IC50 | 3 | — | |
IBRUPFNOCSUECL
|
7.4 | IC50 | 3 | — | |
IZWQPEYVFYWESQ
|
7.4 | IC50 | 3 | — | |
OMLHQPIYXLWGGG
|
7.4 | IC50 | 3 | — | |
PPCFYGSMPQKDDM
|
7.4 | IC50 | 3 | — | |
QCXJZVDATPNNCE
|
7.4 | IC50 | 3 | — | |
SCYDFQIUWZYQDE
|
7.4 | IC50 | 3 | — | |
SFZBPQNERSUWOW
|
7.4 | IC50 | 3 | — |