Target Details
| UniProt AC | P25440 |
|---|---|
| Gene Symbol | BRD2 |
| Protein Name | Bromodomain-containing protein 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 699
- Clinical molecules 0
- Avg pChEMBL 7.25
Active Molecules (699)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HNJGEQPWIDZIRC
|
7.6 | IC50 | 3 | — | |
OGVXCCMPKKUNFP
|
7.6 | IC50 | 3 | — | |
RLAHXCWDADVADO
|
7.6 | IC50 | 4 | — | |
VFDAORCFAAAXRV
|
7.6 | IC50 | 3 | — | |
FDMPGPNYXCYCQJ
|
7.6 | IC50 | 3 | — | |
JSKLBERKQHGHCP
|
7.6 | IC50 | 3 | — | |
RIDHDDTVNQHKEQ
|
7.6 | IC50 | 3 | — | |
DHQSSAHSRGVRJY
|
7.6 | IC50 | 3 | — | |
GQVNARRVGGOXNP
|
7.6 | IC50 | 3 | — | |
GTFJSDPFUPQADT
|
7.6 | IC50 | 2 | — | |
LEMUMFMXNFTRTL
|
7.6 | IC50 | 3 | — | |
POKZINYHLOHGEB
|
7.6 | Kd | 4 | — | |
QLRYSHYUZMZZPY
|
7.6 | IC50 | 4 | — | |
QNOJAPBYTXGBLX
|
7.6 | Ki | 5 | — | |
FUOUPXXFTDVPGM
|
7.5 | IC50 | 3 | — | |
HQEUJXGKBKBFIW
|
7.5 | IC50 | 3 | — | |
KQIUBFKRUFVQEI
|
7.5 | IC50 | 3 | — | |
NRKGWEXMFVBBBE
|
7.5 | IC50 | 3 | — | |
QDMDJWBTMQQUPC
|
7.5 | IC50 | 3 | — | |
RDWRDUFEWMSPGQ
|
7.5 | Kd | 4 | — | |
WCNXRFKEDHKCLC
|
7.5 | IC50 | 3 | — | |
XMRBIQDRTZCVGG
|
7.5 | IC50 | 3 | — | |
GLMGIYSAZNFOHX
|
7.5 | IC50 | 3 | — | |
KVTLTFKBEFZOGC
|
7.5 | IC50 | 3 | — | |
NCLGWTFZOQZNIS
|
7.5 | IC50 | 3 | — | |
NMPGZGXWNHOBFF
|
7.5 | IC50 | 3 | — | |
QUICABMRXTUSBQ
|
7.5 | IC50 | 2 | — | |
UCTNVNGRNJPSOM
|
7.5 | IC50 | 3 | — | |
VLMANYNJKKOADM
|
7.5 | IC50 | 2 | — | |
ZJXAVKZXYZJJKO
|
7.5 | IC50 | 3 | — | |
GTYWOEFUZYKPQR
|
7.5 | IC50 | 3 | — | |
HSMCUAMXZNQLSQ
|
7.5 | IC50 | 3 | — | |
IMXDUOIANVGJIA
|
7.5 | IC50 | 4 | — | |
NAPOLFVZKFHOBG
|
7.5 | IC50 | 4 | — | |
OJCRNHCUTYXXFI
|
7.5 | Kd | 3 | — | |
WQEGQSRMXSLEON
|
7.5 | IC50 | 4 | — | |
IYRDZCVNOKVDNI
|
7.5 | IC50 | 3 | — | |
LORVKFYVSXATKW
|
7.5 | IC50 | 5 | — | |
SNIKOFNWYKITGY
|
7.5 | IC50 | 3 | — | |
SSELZXGQLGXCDT
|
7.5 | IC50 | 3 | — | |
ZZJIAOWVSKZQGQ
|
7.5 | IC50 | 3 | — | |
AIPWZDCZUJGLIF
|
7.5 | IC50 | 3 | — | |
BQDONWPMBNKZCG
|
7.5 | IC50 | 4 | — | |
BYCJBYOKDKPJQP
|
7.5 | IC50 | 3 | — | |
FAPXCSUYTUWYIY
|
7.5 | IC50 | 2 | — | |
FLEGAAQBQHISDY
|
7.5 | IC50 | 3 | — | |
FOEVWVKNXOCNTG
|
7.5 | IC50 | 3 | — | |
HKECFOZBEGKIAX
|
7.5 | IC50 | 3 | — | |
JLNZMTDBARFXJN
|
7.5 | Kd | 9 | — | |
KQIUBFKRUFVQEI
|
7.5 | IC50 | 3 | — |