Target Details
| UniProt AC | P25440 |
|---|---|
| Gene Symbol | BRD2 |
| Protein Name | Bromodomain-containing protein 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17035 (BET) PF00439 (Bromodomain) |
Summary
- Multi-target molecules 699
- Clinical molecules 0
- Avg pChEMBL 7.25
Active Molecules (699)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LRWGLQDVNJOJKQ
|
7.0 | IC50 | 3 | — | |
FNQLTUOQASERQX
|
7.0 | IC50 | 2 | — | |
IXNBIPCXYOBMSS
|
7.0 | IC50 | 3 | — | |
JTXHXYXYGGEYBL
|
7.0 | Kd | 3 | — | |
MWVVALQFXSOQLF
|
7.0 | IC50 | 3 | — | |
NBBLMCRKPAWOPH
|
7.0 | IC50 | 3 | — | |
QIJUHAIEZZEKSX
|
7.0 | IC50 | 3 | — | |
AAFNIAPCKWGXDG
|
7.0 | IC50 | 3 | — | |
BKQJIPRADVVRKL
|
7.0 | IC50 | 3 | — | |
IKGRWYRGRUJEIF
|
7.0 | IC50 | 3 | — | |
OTZHGAAUXLOJFP
|
7.0 | IC50 | 3 | — | |
PVDBPOSKQRWTRG
|
7.0 | IC50 | 3 | — | |
QIJUHAIEZZEKSX
|
7.0 | IC50 | 3 | — | |
XASDFFVVUGREBP
|
7.0 | IC50 | 3 | — | |
AMGMXABLUGQVQD
|
7.0 | IC50 | 3 | — | |
ARWMKZDWGIOCEU
|
7.0 | IC50 | 4 | — | |
BKDMSQCDGPSQFW
|
7.0 | IC50 | 3 | — | |
FAMCYVZRWHZORW
|
7.0 | IC50 | 3 | — | |
FNDFWBANYDEWBA
|
7.0 | Kd | 3 | — | |
HBIBLLVDGBUKCQ
|
7.0 | IC50 | 4 | — | |
IMUJKGKBDBVTGZ
|
7.0 | IC50 | 3 | — | |
JUNKHWUBWMACDY
|
7.0 | IC50 | 3 | — | |
JVAKWUYUZCOCKR
|
7.0 | IC50 | 4 | — | |
NBBLMCRKPAWOPH
|
7.0 | IC50 | 3 | — | |
PXGREUPWZAUELV
|
7.0 | IC50 | 3 | — | |
PXGREUPWZAUELV
|
7.0 | IC50 | 3 | — | |
SSCBXXKTZLTDDN
|
7.0 | IC50 | 3 | — | |
ULIAHCSBBVNLGS
|
7.0 | IC50 | 3 | — | |
XSOFZNARGSJIQN
|
7.0 | IC50 | 4 | — | |
GFDDTDKCZCGJLM
|
7.0 | Kd | 5 | — | |
LMLJGVCFCYGAST
|
7.0 | IC50 | 3 | — | |
RQSRLTLIMDDPDM
|
7.0 | IC50 | 4 | — | |
MTKZUOYFXZHUDU
|
7.0 | IC50 | 3 | — | |
HXVTYKVZGFHITR
|
7.0 | IC50 | 3 | — | |
IMYHVLQAXUTNRG
|
7.0 | IC50 | 3 | — | |
JFPHLFWFVVJKQO
|
7.0 | IC50 | 4 | — | |
OXYDGMKIFXNGOS
|
7.0 | IC50 | 3 | — | |
VLEMFHFORYINCB
|
7.0 | IC50 | 4 | — | |
ALALEIOMSWRNDF
|
7.0 | IC50 | 2 | — | |
AYMBFUSITNSKHY
|
6.9 | IC50 | 3 | — | |
WEQSOZXIXPNDJW
|
6.9 | Kd | 2 | — | |
AREGGTVPTLNTCU
|
6.9 | IC50 | 3 | — | |
BRQOWLMNQSLGPU
|
6.9 | IC50 | 3 | — | |
HXENBKGGEPBXOQ
|
6.9 | IC50 | 3 | — | |
JSJHNZMAOMLIME
|
6.9 | IC50 | 3 | — | |
PIPFCKKGOLUZIH
|
6.9 | IC50 | 3 | — | |
PMIMBFPXSMELLC
|
6.9 | IC50 | 3 | — | |
QXYGIHZVXILREV
|
6.9 | IC50 | 3 | — | |
RTFLOGJKYBGANO
|
6.9 | IC50 | 4 | — | |
SLTHVRXQOKFPLI
|
6.9 | IC50 | 3 | — |