Target Details
| UniProt AC | P25116 |
|---|---|
| Gene Symbol | F2R |
| Protein Name | Proteinase-activated receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 37
- Clinical molecules 0
- Avg pChEMBL 7.26
KEGG Pathways (11)
- Calcium signaling pathway
- Complement and coagulation cascades
- Neuroactive ligand-receptor interaction
- PI3K-Akt signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Phospholipase D signaling pathway
- Platelet activation
- Rap1 signaling pathway
- Regulation of actin cytoskeleton
- cAMP signaling pathway
Active Molecules (37)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LUVNXTSNCPCXQE
|
9.4 | Kd | 2 | — | |
GOQXRFYWUHPILG
|
8.8 | IC50 | 2 | — | |
UEPOSULLGAYZQZ
|
8.7 | IC50 | 2 | — | |
PIRVYNOHTBFSEF
|
8.5 | IC50 | 2 | — | |
QGDLVNWXOJELBV
|
8.5 | IC50 | 2 | — | |
IDEORNGCCVYCFX
|
8.4 | IC50 | 2 | — | |
ZFBVWXYOLVFQGN
|
8.4 | IC50 | 2 | — | |
QJDXGILNNBHQDK
|
8.3 | IC50 | 2 | — | |
YGACWBAYURXDEP
|
7.9 | IC50 | 2 | — | |
FGJKSKYLEOZELA
|
7.7 | IC50 | 3 | — | |
KEDDGIDZMJSBEW
|
7.7 | IC50 | 2 | — | |
XVIKFFNGSSURCJ
|
7.7 | IC50 | 3 | — | |
VNOAMEZLBNKPPP
|
7.6 | IC50 | 2 | — | |
LSKGPGZPROETCR
|
7.5 | IC50 | 2 | — | |
GMPWJHCKUFHLJE
|
7.3 | IC50 | 2 | — | |
FFXFDFRJDPWERF
|
7.2 | IC50 | 2 | — | |
LVCJHIUPGAKASO
|
7.2 | IC50 | 2 | — | |
GZPIECMFJJLDAB
|
7.2 | IC50 | 2 | — | |
AFEBUYQIVROWSL
|
7.1 | IC50 | 3 | — | |
VVKBGBCCSDVWHK
|
7.1 | IC50 | 3 | — | |
ZLWUPXBJIJIQJF
|
7.1 | IC50 | 2 | — | |
BFJWHYCHYOUZLZ
|
7.1 | IC50 | 2 | — | |
CYKYNQSFAYHHEZ
|
7.0 | IC50 | 3 | — | |
LZKMIVXPFPBCFC
|
7.0 | IC50 | 2 | — | |
SRNIWQIVVVDOLO
|
7.0 | IC50 | 2 | — | |
UWNZCZNHUPLBBY
|
6.9 | IC50 | 2 | — | |
BCXNFSKGOXTNLM
|
6.5 | IC50 | 2 | — | |
QOZKFVLJGZGBOI
|
6.5 | IC50 | 3 | — | |
LPHKQDNIANODOF
|
6.3 | IC50 | 2 | — | |
WNSZHTAQLGVRHC
|
6.2 | IC50 | 2 | — | |
YHASTZKIWUZWDO
|
6.2 | IC50 | 2 | — | |
QOZKFVLJGZGBOI
|
6.2 | IC50 | 3 | — | |
XGDVRXHWQGEVTD
|
6.1 | IC50 | 3 | — | |
XGDVRXHWQGEVTD
|
6.1 | IC50 | 3 | — | |
LCFFZUZPPRYCKY
|
6.0 | IC50 | 2 | — | |
VEYNGJJQBIEPNE
|
6.0 | IC50 | 2 | — | |
GUTGOHPTMQPGTD
|
6.0 | IC50 | 3 | — |