Target Details
| UniProt AC | P25105 |
|---|---|
| Gene Symbol | PTAFR |
| Protein Name | Platelet-activating factor receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 16
- Clinical molecules 0
- Avg pChEMBL 6.37
KEGG Pathways (3)
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XNQIOISZPFVUFG
|
7.9 | IC50 | 2 | — | |
DCNXKPFVMNEKDU
|
6.6 | IC50 | 2 | — | |
WDGUBDMXGCFGIL
|
6.6 | IC50 | 2 | — | |
LKFAYNBLUNPUHN
|
6.5 | IC50 | 2 | — | |
DGYJMRJVVGLCDV
|
6.4 | IC50 | 2 | — | |
IIXGCBPDCHNSLC
|
6.4 | IC50 | 2 | — | |
RUAOGLCGDIBHJR
|
6.3 | IC50 | 2 | — | |
OIMUMJMHBPPFFI
|
6.3 | IC50 | 2 | — | |
OCWOTYUFXGGBAW
|
6.2 | IC50 | 2 | — | |
JOFWLTCLBGQGBO
|
6.2 | Ki | 8 | — | |
LQUYEBKTHLMNKY
|
6.2 | IC50 | 2 | — | |
FLTBEMVEAFMWDD
|
6.1 | IC50 | 2 | — | |
OZCVIUHHOUTJJN
|
6.1 | IC50 | 2 | — | |
DKVCJHBRBBPIGM
|
6.0 | IC50 | 2 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
OYMNICOOAXOYPP
|
6.0 | IC50 | 2 | — |