Target Details
| UniProt AC | P25103 |
|---|---|
| Gene Symbol | TACR1 |
| Protein Name | Substance-P receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 589
- Clinical molecules 2
- Avg pChEMBL 8.16
KEGG Pathways (3)
Active Molecules (589)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LCMYTAQFJIXBCQ
|
6.5 | IC50 | 2 | — | |
JVCKKWZCSIKZIY
|
6.5 | IC50 | 2 | — | |
OAVNGCZBHRXUGH
|
6.5 | IC50 | 3 | — | |
JEZKKPXWSVQUPH
|
6.5 | Ki | 3 | — | |
CQJXBNDZWCFOLX
|
6.4 | IC50 | 2 | — | |
ODPRNYGWGVRXIG
|
6.4 | IC50 | 3 | — | |
GDUGRYUTQQIHKS
|
6.4 | IC50 | 2 | — | |
KMXLXHFSSQDIGC
|
6.4 | IC50 | 3 | — | |
BVALXLKHALQQPF
|
6.4 | IC50 | 2 | — | |
XIUWYQPZUOTMGU
|
6.4 | Ki | 2 | — | |
NCJWLSWXMPGOIS
|
6.3 | IC50 | 3 | — | |
PGKXDIMONUAMFR
|
6.3 | Ki | 3 | — | |
BYUMATUURCXQEB
|
6.3 | IC50 | 2 | — | |
DNYAHFKJMPYBQK
|
6.3 | IC50 | 2 | — | |
WAACBTLXCIQAPC
|
6.3 | IC50 | 3 | — | |
WQUXLRVVRRBKCO
|
6.3 | IC50 | 2 | — | |
NHXYSAFTNPANFK
|
6.3 | Ki | 3 | — | |
VVOGLOJOGOEZPO
|
6.2 | IC50 | 2 | — | |
BUBGVFLMAHPWIA
|
6.2 | IC50 | 2 | — | |
HEAUFJZALFKPBA
|
6.2 | Ki | 3 | — | |
HEAUFJZALFKPBA
|
6.2 | Ki | 3 | — | |
SWGQDPWKPYZEEH
|
6.2 | IC50 | 2 | — | |
YQHKVGJQICUJMY
|
6.2 | IC50 | 2 | — | |
FVMGZIMTEZPJGA
|
6.2 | IC50 | 2 | — | |
QKBBGEQUAVGUHW
|
6.2 | Kd | 2 | — | |
UKMJWGFHXMGRNG
|
6.2 | Kd | 2 | — | |
PGKXDIMONUAMFR
|
6.2 | IC50 | 2 | — | |
SIPOLHQPOKEDPH
|
6.2 | IC50 | 2 | — | |
ADXFJIYJEFFOSY
|
6.1 | IC50 | 3 | — | |
MQERJZPDBKDRIH
|
6.1 | IC50 | 2 | — | |
ZLPGKEGAFJLKOK
|
6.1 | IC50 | 3 | — | |
CFDNUNSOUUFTQO
|
6.1 | IC50 | 2 | — | |
YXYOQVJTKQKSTM
|
6.1 | IC50 | 2 | — | |
NFBNIRNKYJTDIE
|
6.1 | IC50 | 16 | Yes | |
AHOUBRCZNHFOSL
|
6.0 | IC50 | 13 | — | |
VIGYJJFBPARTJM
|
6.0 | IC50 | 3 | — | |
VXGPTRVARWWDQI
|
6.0 | IC50 | 2 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
PFOMIAQBONXLRP
|
6.0 | IC50 | 2 | — |