Target Details
| UniProt AC | P25103 |
|---|---|
| Gene Symbol | TACR1 |
| Protein Name | Substance-P receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 589
- Clinical molecules 2
- Avg pChEMBL 8.16
KEGG Pathways (3)
Active Molecules (589)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WMTKHCQGJKXVST
|
12.0 | Ki | 2 | — | |
ADVXLVRKUFJJTA
|
11.6 | Ki | 2 | — | |
ADPQCWUGLGBPRO
|
11.4 | Ki | 2 | — | |
NKULLHQHASCPKR
|
11.4 | Ki | 2 | — | |
PVNAJCHBKOKIIB
|
11.3 | Ki | 2 | — | |
DSXDZHLLPRAKKT
|
11.2 | Ki | 2 | — | |
ZLNYUCXXSDDIFU
|
11.2 | Ki | 3 | — | |
ATJZNASWBNGJGA
|
11.1 | Ki | 2 | — | |
CJYLEVUNMXXSAG
|
11.1 | Ki | 2 | — | |
UTXLSPLKQGPIPL
|
10.9 | IC50 | 2 | — | |
ZGKMSCDQIDVSIK
|
10.8 | Ki | 2 | — | |
CAHGELRDKXVTKA
|
10.6 | IC50 | 2 | — | |
MVWDYFOJQAABRA
|
10.5 | IC50 | 3 | — | |
LVKWUNFNJODDPV
|
10.5 | IC50 | 3 | — | |
VUBAEISRKSELTE
|
10.5 | Ki | 2 | — | |
ZDJFLHCNTGAWQS
|
10.5 | IC50 | 2 | — | |
OIFPROSOIDRACJ
|
10.5 | IC50 | 2 | — | |
VYUZFKRVLLXBRD
|
10.5 | Ki | 2 | — | |
OUYSLNGQLIIZQC
|
10.4 | IC50 | 3 | — | |
XHJXRHNUFXHMEV
|
10.3 | Ki | 2 | — | |
HUBLDDBZWROLJY
|
10.3 | IC50 | 2 | — | |
GVRKQRSTDMXZGX
|
10.3 | Ki | 2 | — | |
ACFPRWCERXMNGY
|
10.3 | Ki | 2 | — | |
DHNLMUQAIWWIEX
|
10.2 | Ki | 2 | — | |
XWNBGDJPEXZSQM
|
10.2 | Ki | 2 | — | |
KTVJZUAZYBDWSQ
|
10.2 | Ki | 2 | — | |
GNFGMQJCVYXXRO
|
10.2 | IC50 | 2 | — | |
CSUAYJZRABTSRO
|
10.1 | IC50 | 2 | — | |
KTIXRTOVKASTTK
|
10.1 | Ki | 2 | — | |
LIXRIEAGLPGVJF
|
10.1 | IC50 | 3 | — | |
ATALOFNDEOCMKK
|
10.1 | IC50 | 3 | — | |
MJOXRJQZLVVZCL
|
10.1 | Ki | 2 | — | |
NUTYWRAIFXRNNI
|
10.1 | IC50 | 2 | — | |
OYKIXMQKLMUJEK
|
10.1 | IC50 | 3 | — | |
PLMUPHYPECRQJW
|
10.0 | IC50 | 3 | — | |
NTYJRAGMLUHRNV
|
10.0 | Ki | 2 | — | |
VBOXQXAJDAUESQ
|
10.0 | IC50 | 2 | — | |
ZOPRZQRKBZNHLP
|
10.0 | Ki | 2 | — | |
ZXJRUKOAFOUFIR
|
10.0 | Ki | 2 | — | |
TWBCIHKYFTWYCV
|
10.0 | Ki | 2 | — | |
PLOFBQMQAHOQHM
|
10.0 | IC50 | 2 | — | |
SJHZTGDJTIZMSK
|
10.0 | Ki | 3 | — | |
IPMMBNAOLDMKAM
|
9.9 | IC50 | 2 | — | |
IQGTUPXJLRMAOA
|
9.9 | Ki | 2 | — | |
OXXARYIRJZWVPQ
|
9.9 | Ki | 2 | — | |
GXIFPPFQXPIEKY
|
9.9 | IC50 | 2 | — | |
CYKFSGXEZOAASR
|
9.9 | IC50 | 2 | — | |
VHQVJYKYAGBACO
|
9.8 | Ki | 3 | — | |
ZIWFCOIGUNPHPM
|
9.8 | IC50 | 5 | — | |
OEIZZOMBDHTIGH
|
9.8 | IC50 | 2 | — |