Target Details
| UniProt AC | P25101 |
|---|---|
| Gene Symbol | EDNRA |
| Protein Name | Endothelin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 535
- Clinical molecules 0
- Avg pChEMBL 8.16
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (535)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QDRPQGXYQQITQV
|
7.4 | Ki | 2 | — | |
JMWQBPRIANCZRQ
|
7.3 | IC50 | 2 | — | |
UPQGVXBBBKNPNZ
|
7.3 | IC50 | 2 | — | |
UVTGPXVPTNTUDR
|
7.3 | Ki | 2 | — | |
AIVZWVQMNJFOIL
|
7.3 | IC50 | 2 | — | |
BYBPPGGQNVVISN
|
7.3 | IC50 | 2 | — | |
FDVBFLHJYUCEKU
|
7.3 | IC50 | 2 | — | |
GCISLFODTRCVKS
|
7.3 | IC50 | 2 | — | |
JPRDUKLJMTUKCJ
|
7.3 | IC50 | 2 | — | |
RBIUYHJGRUEIPU
|
7.3 | IC50 | 2 | — | |
GWVRRZASHHOARI
|
7.3 | IC50 | 2 | — | |
MSRYVIMFULZUGC
|
7.3 | Ki | 2 | — | |
RGQAYSMKTZIBMN
|
7.3 | IC50 | 2 | — | |
XUMJJSAQQCTKAO
|
7.3 | IC50 | 3 | — | |
GWBCKOWLDKFIHO
|
7.3 | IC50 | 2 | — | |
NQDCDWVUSPOECA
|
7.3 | IC50 | 2 | — | |
ZHWQNJCSTDEVGM
|
7.3 | IC50 | 2 | — | |
FPZOGKSKYWZFIO
|
7.3 | IC50 | 2 | — | |
KZOKREKJZZEWAD
|
7.3 | IC50 | 2 | — | |
SGMHXYMWOLAIMX
|
7.3 | IC50 | 2 | — | |
PZBNHZOXFOMEDO
|
7.3 | Ki | 2 | — | |
XMLFZKYJSPXNGH
|
7.2 | IC50 | 2 | — | |
AVUMTAXWDOUGCR
|
7.2 | IC50 | 2 | — | |
OVPKPOGJHFVIFR
|
7.2 | IC50 | 2 | — | |
KEGRAIQJSRYPGR
|
7.2 | IC50 | 2 | — | |
MOTJMGVDPWRKOC
|
7.2 | Ki | 2 | — | |
WYLRXEBBERTKHN
|
7.2 | IC50 | 2 | — | |
ASUNSLBCCFVKJD
|
7.2 | IC50 | 2 | — | |
FDDMPZZHBROSPE
|
7.2 | IC50 | 2 | — | |
QLKHVLXMFAFDAZ
|
7.2 | IC50 | 2 | — | |
BYCLKBXHEZQIHD
|
7.2 | IC50 | 2 | — | |
HEGRKFSINVTUKI
|
7.1 | IC50 | 2 | — | |
HDHCADXZMJNZJH
|
7.1 | IC50 | 2 | — | |
NHKDLOQLHLFRRT
|
7.1 | IC50 | 2 | — | |
YLMSOIIFAYJNMX
|
7.1 | IC50 | 2 | — | |
LYOPDHNZJQBGAC
|
7.1 | IC50 | 2 | — | |
HQIPFADRUMZDIT
|
7.1 | IC50 | 2 | — | |
NIGCNIFGPYTDPJ
|
7.1 | IC50 | 2 | — | |
UJGUMHQLVYROSG
|
7.1 | Ki | 2 | — | |
QSFFFSPNGBKTGJ
|
7.1 | IC50 | 2 | — | |
XBXUZKKIOMHQDF
|
7.1 | IC50 | 2 | — | |
YTNUBEUYCFIHBS
|
7.1 | IC50 | 2 | — | |
HDWHUKBOFNHSSO
|
7.1 | IC50 | 2 | — | |
CFTTVXIBXXPWEU
|
7.1 | Ki | 2 | — | |
KKGSEDUFHOPCFO
|
7.0 | IC50 | 2 | — | |
FFXSFOBUYYTLRH
|
7.0 | IC50 | 2 | — | |
OTMGLEOGWQJHIQ
|
7.0 | IC50 | 2 | — | |
TWBVBLFAEWNYQQ
|
7.0 | IC50 | 2 | — | |
GBYVJKRBUNPVLB
|
7.0 | IC50 | 2 | — | |
IISLJISTBMPEAA
|
7.0 | IC50 | 2 | — |