Target Details
| UniProt AC | P25101 |
|---|---|
| Gene Symbol | EDNRA |
| Protein Name | Endothelin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 535
- Clinical molecules 0
- Avg pChEMBL 8.16
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (535)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WUYGPPAFDHJCRQ
|
7.7 | IC50 | 2 | — | |
DNIIBGYNGASUDE
|
7.7 | IC50 | 2 | — | |
GQTAIGFWINAVHA
|
7.7 | IC50 | 2 | — | |
SCMXLDCMGHKGGU
|
7.7 | IC50 | 2 | — | |
PMUCOFCFESYTCH
|
7.7 | Ki | 2 | — | |
NHVWTLKWIKMKNS
|
7.7 | IC50 | 2 | — | |
TVTJICVMTXUAKS
|
7.7 | IC50 | 2 | — | |
NNXCMHJFFYTMCA
|
7.7 | IC50 | 2 | — | |
AEDJOIBTFWFFLB
|
7.7 | IC50 | 2 | — | |
GAICYMPBDZVZOU
|
7.7 | IC50 | 2 | — | |
KZSPAFPPOAOZPK
|
7.7 | IC50 | 2 | — | |
BEGQGXHBEYDHFL
|
7.6 | IC50 | 2 | — | |
OCZIRSIFHBBDKN
|
7.6 | Ki | 2 | — | |
IGKCOJUPPUGBIE
|
7.6 | IC50 | 2 | — | |
GZABEWFFPRCWQI
|
7.6 | IC50 | 2 | — | |
NTQWAQFOJQQOTK
|
7.6 | IC50 | 3 | — | |
SIPPOBLYWAIKGU
|
7.6 | IC50 | 2 | — | |
WQLXYQSKSGEIPU
|
7.6 | IC50 | 4 | — | |
YNFUBOJUAKNKLF
|
7.6 | IC50 | 2 | — | |
FQXLGGFHDJJJJO
|
7.6 | IC50 | 2 | — | |
FRQPGCPVRMZTNE
|
7.6 | IC50 | 2 | — | |
PUEQTWGTNQUURY
|
7.6 | IC50 | 2 | — | |
QWDHLTWAAVZDIR
|
7.6 | Ki | 2 | — | |
BZSLFEJGVQKVKX
|
7.6 | IC50 | 2 | — | |
PFRXWKQQCRIVDP
|
7.6 | IC50 | 2 | — | |
HTNBCWLAXCOARB
|
7.6 | IC50 | 2 | — | |
LUQZWCBOERIKEO
|
7.5 | IC50 | 2 | — | |
NVONIBWWXNXALH
|
7.5 | IC50 | 2 | — | |
BOQQYCYLUTYLGS
|
7.5 | IC50 | 2 | — | |
KRSWVPASAJDUGK
|
7.5 | IC50 | 2 | — | |
VVOGFCYZFAKNMH
|
7.5 | IC50 | 2 | — | |
WCPSMXYWDQGMJD
|
7.5 | IC50 | 2 | — | |
XJSUBSFOTRRUES
|
7.5 | IC50 | 2 | — | |
GBDHMDQPXDYBRO
|
7.5 | IC50 | 2 | — | |
ZHXNJGISXVIIND
|
7.5 | Ki | 2 | — | |
VJGDGBUWSOZGFC
|
7.5 | Ki | 2 | — | |
FTHTWZGSLVJZJB
|
7.5 | Ki | 2 | — | |
KNUFDNSKLOOTIB
|
7.5 | IC50 | 2 | — | |
OSRCBCUYZBTKBZ
|
7.5 | IC50 | 2 | — | |
QPUBINGNDLKIHN
|
7.5 | IC50 | 2 | — | |
XPUJKHFCHQYTEQ
|
7.5 | IC50 | 2 | — | |
DTDRDEIFMKNNTL
|
7.5 | IC50 | 2 | — | |
BQFWUVDRXODPBL
|
7.4 | IC50 | 2 | — | |
FKUFTGMFORIVAP
|
7.4 | IC50 | 2 | — | |
IKSWGOKQGJQKIW
|
7.4 | IC50 | 2 | — | |
JGAUQCSCABMOTB
|
7.4 | IC50 | 2 | — | |
NNGHGYQUGDQKJY
|
7.4 | IC50 | 2 | — | |
UTSWGARHIRATMS
|
7.4 | Ki | 2 | — | |
GJPICJJJRGTNOD
|
7.4 | IC50 | 2 | — | |
XYHBLDIJAJYURE
|
7.4 | Ki | 2 | — |