Target Details
| UniProt AC | P25101 |
|---|---|
| Gene Symbol | EDNRA |
| Protein Name | Endothelin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 535
- Clinical molecules 0
- Avg pChEMBL 8.16
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (535)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MIPNODJPKTVQHX
|
8.0 | IC50 | 2 | — | |
UPRKHNRGBDTKKR
|
8.0 | IC50 | 2 | — | |
QCHYZDXDWZKACW
|
8.0 | IC50 | 2 | — | |
UMVOCHGUCRDMRD
|
8.0 | IC50 | 2 | — | |
VAXUKYCSAUELNZ
|
8.0 | IC50 | 2 | — | |
KQTXBXFCFQJGGY
|
8.0 | IC50 | 2 | — | |
MZAAFBAXCKYSNN
|
8.0 | IC50 | 2 | — | |
VACPWIZSMORWDJ
|
8.0 | IC50 | 2 | — | |
JNUYVBGNCBJGHQ
|
7.9 | IC50 | 2 | — | |
FINMPMBYTTVLPJ
|
7.9 | IC50 | 2 | — | |
PQJLYRULHJYQDW
|
7.9 | IC50 | 2 | — | |
UJPMGYUNKDMJEA
|
7.9 | IC50 | 2 | — | |
GUILESAVAVIDIH
|
7.9 | Ki | 2 | — | |
JKNAAXSOIGHTLX
|
7.9 | IC50 | 2 | — | |
SXEVCCXWQGAXSQ
|
7.9 | IC50 | 2 | — | |
XDNAXXIOBHFZDQ
|
7.9 | IC50 | 2 | — | |
XSAFCBSWMREXMT
|
7.9 | IC50 | 2 | — | |
HFWWOBMAMIJJEP
|
7.9 | IC50 | 2 | — | |
WAOUMQDGIOSVAF
|
7.9 | IC50 | 2 | — | |
XIKMSNPORKHQQQ
|
7.9 | IC50 | 2 | — | |
BCRJIIJVFJJYRD
|
7.8 | IC50 | 2 | — | |
CMPCSJBKUBWQGQ
|
7.8 | IC50 | 2 | — | |
JBRKIZWDQQOPCK
|
7.8 | Ki | 2 | — | |
SWIPVSPLUXWKTL
|
7.8 | IC50 | 2 | — | |
XPOWMKNHKCJZNA
|
7.8 | IC50 | 2 | — | |
ZLSUWQHIYSFEQP
|
7.8 | IC50 | 2 | — | |
APXDEEHRWJDGMC
|
7.8 | IC50 | 2 | — | |
BJSXTKDRYZUWEL
|
7.8 | Ki | 2 | — | |
JPBZOZDHBRRLBM
|
7.8 | IC50 | 2 | — | |
UIYNSXMUJGBENK
|
7.8 | IC50 | 2 | — | |
VGWWIMUJYACUED
|
7.8 | IC50 | 2 | — | |
BKGYGEADRLJUHK
|
7.8 | IC50 | 2 | — | |
DUZPNAKTFLDXQA
|
7.8 | IC50 | 2 | — | |
QPZJVKVINGMRAL
|
7.8 | IC50 | 2 | — | |
UHXUKJPNFOYGKB
|
7.8 | IC50 | 2 | — | |
XDNAXXIOBHFZDQ
|
7.8 | IC50 | 2 | — | |
AXVBSGVXXMZTEC
|
7.8 | IC50 | 2 | — | |
FHRCXZSDINFQMI
|
7.8 | IC50 | 2 | — | |
GEKLWHMKKGCLLE
|
7.8 | IC50 | 2 | — | |
HOULTIREPNOFQE
|
7.8 | IC50 | 2 | — | |
PBTTZSSLQDEUPI
|
7.8 | IC50 | 2 | — | |
XAJNNLNUOAQGQO
|
7.8 | IC50 | 2 | — | |
SDXSGUVLSFVWRF
|
7.8 | IC50 | 2 | — | |
TWGYPFLCDZVWJV
|
7.8 | IC50 | 2 | — | |
CQHLNCPJLNXFBC
|
7.8 | IC50 | 2 | — | |
CKAWNKDSMUUPOR
|
7.7 | IC50 | 2 | — | |
KEZZZBNAPVGBEW
|
7.7 | IC50 | 2 | — | |
TUYWTLTWNJOZNY
|
7.7 | IC50 | 2 | — | |
VXJUFLPIZFIKQL
|
7.7 | IC50 | 2 | — | |
WFGXYWSSRLHSJI
|
7.7 | IC50 | 2 | — |