Target Details
| UniProt AC | P25101 |
|---|---|
| Gene Symbol | EDNRA |
| Protein Name | Endothelin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 535
- Clinical molecules 0
- Avg pChEMBL 8.16
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (535)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DVNMKMKQUAYZDJ
|
8.2 | IC50 | 2 | — | |
FZNWHURKGWXPCC
|
8.2 | IC50 | 2 | — | |
MHNJEAOUFUNYKE
|
8.2 | IC50 | 2 | — | |
SEXZWLMIBXVFQM
|
8.2 | IC50 | 2 | — | |
YFGVPMLVIXUCGP
|
8.2 | IC50 | 2 | — | |
FYULQKSAMXDPLJ
|
8.2 | Ki | 2 | — | |
LSQXFROVPNDBMN
|
8.2 | IC50 | 2 | — | |
TUTZGEFUGWQBKP
|
8.2 | IC50 | 2 | — | |
VIVHYWNEMYNSTR
|
8.2 | IC50 | 2 | — | |
FREUSOYKQUIGQQ
|
8.2 | Ki | 2 | — | |
JOZGLYQYYYGZBS
|
8.2 | IC50 | 2 | — | |
MNJMLQKJRCXWRC
|
8.2 | Ki | 2 | — | |
MRZPJCAABGPJED
|
8.2 | IC50 | 2 | — | |
PWHUJWODHSRAIM
|
8.2 | IC50 | 2 | — | |
UGJAKYVVBJWFEZ
|
8.2 | IC50 | 2 | — | |
VTCDHOQFPYTIFV
|
8.2 | IC50 | 2 | — | |
FGGUYHAUIAJAKH
|
8.1 | IC50 | 2 | — | |
GEAANMFRDZRIIE
|
8.1 | IC50 | 2 | — | |
QWIJRDPSRHJFIY
|
8.1 | IC50 | 2 | — | |
MHZFPYMEACEGKL
|
8.1 | IC50 | 2 | — | |
AUSMSARLDRBCDW
|
8.1 | IC50 | 2 | — | |
WLXMNQFBLVMITG
|
8.1 | IC50 | 2 | — | |
YOMSYVFQYBPECD
|
8.1 | IC50 | 2 | — | |
CFOMGVYXSNFELK
|
8.1 | IC50 | 2 | — | |
ASYDIUHFIWWNJR
|
8.1 | IC50 | 2 | — | |
HZWIXRSMTHDZGL
|
8.1 | IC50 | 2 | — | |
IAHNMFPHUACREU
|
8.1 | Ki | 2 | — | |
MAJFWFWHJWCHLH
|
8.1 | IC50 | 2 | — | |
MOXPGMJEOXCNPF
|
8.1 | IC50 | 2 | — | |
VEMZPXZQLOLLKQ
|
8.1 | IC50 | 2 | — | |
WSNWXTKIOPWVDW
|
8.1 | IC50 | 2 | — | |
CQHSRRONBVIJRO
|
8.1 | IC50 | 2 | — | |
KPISXONXINCUAB
|
8.1 | IC50 | 2 | — | |
OBNJEEOFTPJHQY
|
8.1 | IC50 | 2 | — | |
QLRLGCLZQTWZOK
|
8.1 | Ki | 2 | — | |
NSVNTHSZOXQBPE
|
8.1 | IC50 | 2 | — | |
PGAMLYVKCIXYNX
|
8.1 | IC50 | 2 | — | |
ITICTHRGYDERJA
|
8.1 | IC50 | 2 | — | |
ZYPQETRCACBJNS
|
8.1 | IC50 | 2 | — | |
KIJALYSAGLYTQO
|
8.0 | IC50 | 2 | — | |
SQHUBOCKWBVIDO
|
8.0 | IC50 | 2 | — | |
WETZUHODUGXVKY
|
8.0 | Ki | 2 | — | |
OGTVYDGVOOLHDI
|
8.0 | IC50 | 2 | — | |
QLOACGMSZNOMDZ
|
8.0 | IC50 | 2 | — | |
WRFHGDPIDHPWIQ
|
8.0 | Ki | 2 | — | |
BYIKTFONIZDLEI
|
8.0 | IC50 | 2 | — | |
CIMUQXQFDACEAW
|
8.0 | Ki | 2 | — | |
CTANMDRPZQDKDO
|
8.0 | IC50 | 2 | — | |
GKCAKABSOVLWHG
|
8.0 | IC50 | 2 | — | |
GVIAAZGPMZKJBY
|
8.0 | IC50 | 2 | — |