Target Details
| UniProt AC | P25101 |
|---|---|
| Gene Symbol | EDNRA |
| Protein Name | Endothelin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 535
- Clinical molecules 0
- Avg pChEMBL 8.16
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (535)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VWXMUZZYWKEWJY
|
8.5 | Ki | 2 | — | |
NSROWKBSRVFCCQ
|
8.4 | IC50 | 2 | — | |
RQKVNFYBHIQIDV
|
8.4 | IC50 | 2 | — | |
VUAQGALNRBYHNG
|
8.4 | IC50 | 2 | — | |
JQAHCXASBUTBKC
|
8.4 | IC50 | 2 | — | |
KOWYKBJZTIDYKI
|
8.4 | Ki | 2 | — | |
MRBWXOFHOJHYOZ
|
8.4 | IC50 | 2 | — | |
FYQSINZSEYBXAC
|
8.4 | Kd | 2 | — | |
HRAQSWKGRRUBDJ
|
8.4 | IC50 | 2 | — | |
JZVDVZMUHGSKGI
|
8.4 | IC50 | 2 | — | |
QGSBCBLFBNGHAE
|
8.4 | IC50 | 2 | — | |
YDIGUOCUKLHGNZ
|
8.4 | IC50 | 2 | — | |
RXNZJEAMURXNLG
|
8.4 | IC50 | 2 | — | |
CBJKZXKXUSTFHL
|
8.4 | IC50 | 2 | — | |
YPXSZXRASAVIKK
|
8.4 | IC50 | 2 | — | |
XIIITWQEAPOZLF
|
8.3 | IC50 | 2 | — | |
GMNFTSXERCOCMB
|
8.3 | IC50 | 2 | — | |
VRSKDQFILRKSHK
|
8.3 | IC50 | 2 | — | |
BOZMVLDNYMRJIR
|
8.3 | IC50 | 2 | — | |
LZMBWESXCWUQBJ
|
8.3 | IC50 | 2 | — | |
VVGRGSRZVVXEEN
|
8.3 | Ki | 2 | — | |
GJEGFKNDKHXDSQ
|
8.3 | Ki | 2 | — | |
LGRQZNNALZAMDJ
|
8.3 | Ki | 2 | — | |
RXNZJEAMURXNLG
|
8.3 | IC50 | 2 | — | |
XRUKXLWYVUMZLF
|
8.3 | Ki | 2 | — | |
KANHASGBLWIAIA
|
8.3 | IC50 | 2 | — | |
MWHGEJXLFJLVHX
|
8.3 | Ki | 2 | — | |
ACMPQUAKYNONQE
|
8.2 | IC50 | 2 | — | |
GGEVZGHUELFPFK
|
8.2 | IC50 | 2 | — | |
BKUCZUUARYQRPP
|
8.2 | IC50 | 2 | — | |
FEJVSJIALLTFRP
|
8.2 | Ki | 2 | — | |
FEJVSJIALLTFRP
|
8.2 | Ki | 2 | — | |
FEJVSJIALLTFRP
|
8.2 | Ki | 2 | — | |
HVBUELUOUQXXRH
|
8.2 | Ki | 2 | — | |
NNLKMQXTQXTMET
|
8.2 | IC50 | 2 | — | |
NPLNAUBFRRXHRY
|
8.2 | Ki | 2 | — | |
RZTQQRCQEYQARM
|
8.2 | IC50 | 2 | — | |
YCVDVWIZRUNCFR
|
8.2 | IC50 | 2 | — | |
YLJHCAFDKWQJPI
|
8.2 | IC50 | 2 | — | |
UZLLGNWABVRSKB
|
8.2 | IC50 | 2 | — | |
DWRQMVBEIBBSTC
|
8.2 | IC50 | 2 | — | |
FYPZYGLVQHCNCC
|
8.2 | IC50 | 2 | — | |
HTKNCJNRSZJTJH
|
8.2 | IC50 | 2 | — | |
LZBDEPUGFFURHL
|
8.2 | IC50 | 2 | — | |
LZPJHRAWMATYTH
|
8.2 | IC50 | 2 | — | |
MNJJBWIQROUNDM
|
8.2 | IC50 | 2 | — | |
NEOVBIIJKPUROI
|
8.2 | Ki | 2 | — | |
WYPXYGWFNRNTHH
|
8.2 | IC50 | 2 | — | |
PQGJCQZVHZMJFI
|
8.2 | IC50 | 2 | — | |
ADOZPFPWNPYHGT
|
8.2 | IC50 | 2 | — |