Target Details
| UniProt AC | P25101 |
|---|---|
| Gene Symbol | EDNRA |
| Protein Name | Endothelin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 535
- Clinical molecules 0
- Avg pChEMBL 8.16
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (535)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FHOLSLVTQPRBKJ
|
8.7 | IC50 | 2 | — | |
JKISBSRHDYZOEO
|
8.7 | Ki | 2 | — | |
MNRPBSOBVCAVNX
|
8.7 | IC50 | 2 | — | |
NBDFXMDYBLSGLX
|
8.7 | Ki | 2 | — | |
XYZWCNYWABHTRK
|
8.7 | IC50 | 2 | — | |
PYQNCKSTTLEMCS
|
8.7 | Ki | 2 | — | |
AQDCZLZCKZWUCZ
|
8.7 | IC50 | 2 | — | |
KSGHGYRWLMKYNA
|
8.7 | IC50 | 2 | — | |
KWXXXHXCVVFIMQ
|
8.7 | Ki | 2 | — | |
RPBOIJRVAJKCSF
|
8.7 | IC50 | 2 | — | |
SBPQWNOPLSRSMS
|
8.7 | Ki | 2 | — | |
SQHRONMOLLICCQ
|
8.7 | IC50 | 2 | — | |
CROFEMTXJUXGTE
|
8.7 | IC50 | 2 | — | |
QYVHDIUYFHTCJX
|
8.7 | IC50 | 2 | — | |
YBWLTKFZAOSWSM
|
8.7 | IC50 | 2 | — | |
CLSJNXXMIVKULC
|
8.7 | Ki | 2 | — | |
DEOGRJUDPLWPSR
|
8.7 | IC50 | 2 | — | |
HAIMYEQNXQUSSG
|
8.7 | IC50 | 2 | — | |
HUDYDAYXYKCRPT
|
8.7 | Ki | 2 | — | |
PGAMLYVKCIXYNX
|
8.7 | IC50 | 2 | — | |
MMVFGIYZPKSYRV
|
8.6 | Ki | 2 | — | |
MWZFOVILFVOLMJ
|
8.6 | IC50 | 2 | — | |
AIJJGHXRGHAKEG
|
8.6 | IC50 | 2 | — | |
IDRSXRPOEONBKT
|
8.6 | IC50 | 2 | — | |
NKONTEUZTOHVNH
|
8.6 | IC50 | 2 | — | |
OOUHAJURRQCGRG
|
8.6 | Ki | 2 | — | |
BSUWUKYJNUNGOM
|
8.6 | IC50 | 2 | — | |
GDAGOGOXJLUVGB
|
8.6 | IC50 | 2 | — | |
MHHROYOBQSBUEV
|
8.6 | IC50 | 2 | — | |
BSLISXSHQLGIIZ
|
8.6 | IC50 | 2 | — | |
RJXHHVXIVAHBHS
|
8.6 | IC50 | 2 | — | |
XBKVYIJFYBIMJN
|
8.5 | Ki | 2 | — | |
BTPMMVWQHRCMQR
|
8.5 | IC50 | 2 | — | |
DEYKKRWFIMYKJM
|
8.5 | IC50 | 2 | — | |
KXJZFAQLRGGYSV
|
8.5 | IC50 | 2 | — | |
YJGADOCQUFXVMH
|
8.5 | IC50 | 2 | — | |
ZQMGLMDAJMDRHF
|
8.5 | IC50 | 2 | — | |
FJHPXCQTPSEFDQ
|
8.5 | IC50 | 2 | — | |
KBYIOWQONLGJJU
|
8.5 | Ki | 2 | — | |
RDFPZCGBCKZXNO
|
8.5 | IC50 | 2 | — | |
WUNUEBZYLIUGHH
|
8.5 | Ki | 2 | — | |
DAZOXLCENQFWSQ
|
8.5 | IC50 | 2 | — | |
OYGNCRBWGRCEDM
|
8.5 | IC50 | 2 | — | |
HLYUXTAHAPGOGF
|
8.5 | IC50 | 2 | — | |
DKULOVKANLVDEA
|
8.5 | IC50 | 2 | — | |
KSWCYNIYGNMXLW
|
8.5 | IC50 | 2 | — | |
CLSJNXXMIVKULC
|
8.5 | Ki | 2 | — | |
LFVLYJPEMPWXGS
|
8.5 | IC50 | 2 | — | |
LTFMLNPARFSYNA
|
8.5 | IC50 | 2 | — | |
PYSZMARKHQLZJY
|
8.5 | IC50 | 2 | — |