Target Details
| UniProt AC | P25101 |
|---|---|
| Gene Symbol | EDNRA |
| Protein Name | Endothelin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 535
- Clinical molecules 0
- Avg pChEMBL 8.16
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (535)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HEEXATKNWQMTKJ
|
9.1 | IC50 | 2 | — | |
OQVTWUJKWGKZHT
|
9.1 | Ki | 2 | — | |
VLHPYESMRDUJNS
|
9.1 | Ki | 2 | — | |
DTXFUEYWZXGNEF
|
9.0 | IC50 | 2 | — | |
FCGUSVKFZTVUQB
|
9.0 | IC50 | 2 | — | |
ITRTVLHSTSAZIL
|
9.0 | IC50 | 2 | — | |
NDGMTIKKHLLDIV
|
9.0 | IC50 | 2 | — | |
NONLTBWVEZEZFY
|
9.0 | IC50 | 2 | — | |
OUJTZYPIHDYQMC
|
9.0 | IC50 | 2 | — | |
OUJTZYPIHDYQMC
|
9.0 | Ki | 2 | — | |
PBFKMRLPTUCFLU
|
9.0 | IC50 | 2 | — | |
PIWOCJNYDKRQRS
|
9.0 | IC50 | 2 | — | |
WBTXDANWVHPDGU
|
9.0 | IC50 | 2 | — | |
ZWURMMRAUYXFRY
|
9.0 | IC50 | 2 | — | |
GLCKXJLCYIJMRB
|
9.0 | Ki | 2 | — | |
JHOHFSMURHXTHA
|
9.0 | IC50 | 2 | — | |
JOBIZVVLDQEHKD
|
9.0 | IC50 | 2 | — | |
KVMLOIHJNDCBKI
|
9.0 | IC50 | 2 | — | |
XSSAXXJNGRXQCR
|
9.0 | IC50 | 2 | — | |
KJNXTLHIZCKQRF
|
8.9 | IC50 | 2 | — | |
OXHAHXSAOMBNOX
|
8.9 | IC50 | 2 | — | |
SCOBRKBPUKEATJ
|
8.9 | IC50 | 2 | — | |
FWIARXJRYJCABB
|
8.9 | IC50 | 2 | — | |
HAHANBGRLRTDGL
|
8.9 | Ki | 2 | — | |
OZRQEMUTNMRJTM
|
8.9 | IC50 | 2 | — | |
WZCUCQGZYXGPHF
|
8.9 | Ki | 2 | — | |
ADKWUFCPMCLUKI
|
8.8 | IC50 | 2 | — | |
JOFLWUQNEHCQRX
|
8.8 | IC50 | 2 | — | |
OXPNVLRJIHCUBM
|
8.8 | IC50 | 2 | — | |
PHWXUGHIIBDVKD
|
8.8 | IC50 | 2 | — | |
RULBFQDDCRBSBY
|
8.8 | IC50 | 2 | — | |
SENIALTXHXJCNY
|
8.8 | IC50 | 2 | — | |
VNLAEVZRIYGZCY
|
8.8 | IC50 | 2 | — | |
ZXSBLFBQTHAAHA
|
8.8 | IC50 | 2 | — | |
JNFNRBRGVCBLHK
|
8.8 | Ki | 2 | — | |
QRKZNZMLWQPCPE
|
8.8 | IC50 | 2 | — | |
UTSKZBKTKROJBZ
|
8.8 | IC50 | 2 | — | |
FZJJZYJWWWMPOB
|
8.8 | IC50 | 2 | — | |
VIQIKJNRAFJKTQ
|
8.8 | IC50 | 2 | — | |
YZQQVZQBQWFHTP
|
8.8 | IC50 | 2 | — | |
IFLIQLQVUMXNFU
|
8.8 | Ki | 2 | — | |
KAAWXPGZQHJMQL
|
8.8 | IC50 | 2 | — | |
ARFNEXZBRRNUKE
|
8.8 | IC50 | 2 | — | |
BRSITRUZDCGGKH
|
8.8 | IC50 | 2 | — | |
DJUNTHAWPBMJGJ
|
8.8 | IC50 | 2 | — | |
IDINHRPVYGDPHV
|
8.8 | IC50 | 2 | — | |
ARCCNAPMMHWOCU
|
8.7 | IC50 | 2 | — | |
NMXUCISAFBDZIZ
|
8.7 | IC50 | 2 | — | |
PUMKVXYNDYQHJI
|
8.7 | IC50 | 2 | — | |
CSBNIDOCJNQVQX
|
8.7 | Ki | 2 | — |