Target Details
| UniProt AC | P25101 |
|---|---|
| Gene Symbol | EDNRA |
| Protein Name | Endothelin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 535
- Clinical molecules 0
- Avg pChEMBL 8.16
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (535)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IPZKGERDMRMXJO
|
9.7 | IC50 | 2 | — | |
XBXKAPLYGJALOL
|
9.7 | IC50 | 2 | — | |
AQEWYBHXBBBFNY
|
9.7 | IC50 | 2 | — | |
XNGPPJRUZXMHOV
|
9.7 | IC50 | 2 | — | |
HAHANBGRLRTDGL
|
9.6 | IC50 | 2 | — | |
BMNFTWGABWKVKN
|
9.5 | IC50 | 2 | — | |
FAYAMAAFPRXGJT
|
9.5 | IC50 | 2 | — | |
IUTFNAAZZLIBQX
|
9.5 | IC50 | 2 | — | |
OOJYMKAJOJBARX
|
9.5 | IC50 | 2 | — | |
PWIPORDFWDZCJG
|
9.5 | IC50 | 2 | — | |
XYKNJZNFEGDDIP
|
9.5 | IC50 | 2 | — | |
OFCTYBMKKTVKCR
|
9.5 | Ki | 2 | — | |
BFGUYLRYXCFHGG
|
9.5 | IC50 | 2 | — | |
JMCMZOQWXJPCLI
|
9.4 | IC50 | 2 | — | |
FPJPMEXULUCUCB
|
9.4 | Ki | 2 | — | |
FYDHNMUVDRWWCO
|
9.4 | IC50 | 2 | — | |
HMBISNTYKZVPJD
|
9.4 | Ki | 2 | — | |
MIOQPXBHUMVZRF
|
9.4 | IC50 | 2 | — | |
YAWNVAQKVARTGQ
|
9.4 | IC50 | 2 | — | |
YPBPZJHPGUUGME
|
9.4 | IC50 | 2 | — | |
UUAVCCWBNUITBB
|
9.4 | Ki | 2 | — | |
UUAVCCWBNUITBB
|
9.4 | Ki | 2 | — | |
BATSJXIVNKJCKQ
|
9.3 | IC50 | 2 | — | |
MXLGWPUNPPHJQC
|
9.3 | IC50 | 2 | — | |
LFWCJABOXHSRGC
|
9.3 | IC50 | 2 | — | |
GHIWIAMAJCWXDD
|
9.3 | Ki | 2 | — | |
ABTJDYUDDLHWCG
|
9.3 | IC50 | 2 | — | |
JGCMEBMXRHSZKX
|
9.3 | IC50 | 3 | — | |
TYLZGSIGPRVNQJ
|
9.3 | IC50 | 2 | — | |
UTGRGVUJLJJKSH
|
9.3 | IC50 | 2 | — | |
ZWTAXWXITAZUQP
|
9.3 | IC50 | 2 | — | |
ILKUULNNGMUWFG
|
9.3 | IC50 | 2 | — | |
AEDZVHIKLJEHDR
|
9.3 | IC50 | 2 | — | |
JOMWRKGBRATICM
|
9.3 | IC50 | 2 | — | |
UEHPBBFVUYURNP
|
9.3 | IC50 | 2 | — | |
YGARCWJUVOXSDS
|
9.2 | IC50 | 2 | — | |
YCDUZUIVJLJHQL
|
9.2 | IC50 | 2 | — | |
BIHSQJMJRJBBHK
|
9.2 | IC50 | 2 | — | |
DASGRKPWAFYAFD
|
9.2 | IC50 | 2 | — | |
GADXZXTXFHEOKH
|
9.2 | IC50 | 2 | — | |
KYDWTWOSIICWFQ
|
9.2 | Ki | 2 | — | |
YNKZURRWQXRKDP
|
9.2 | IC50 | 2 | — | |
IGUNGSMXNZWMPG
|
9.1 | IC50 | 2 | — | |
ICAHNKLYQDWFQQ
|
9.1 | IC50 | 2 | — | |
MODHKIOUVGRQCC
|
9.1 | IC50 | 2 | — | |
PIJUSICWAKBTEZ
|
9.1 | IC50 | 2 | — | |
PYNCHZOAMKYGTR
|
9.1 | IC50 | 2 | — | |
BSMQWDCPKODFQI
|
9.1 | IC50 | 2 | — | |
JDIFCWUHBJXZLK
|
9.1 | IC50 | 2 | — | |
NRDKXLWFPVYSKL
|
9.1 | IC50 | 2 | — |