Target Details
| UniProt AC | P25101 |
|---|---|
| Gene Symbol | EDNRA |
| Protein Name | Endothelin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 535
- Clinical molecules 0
- Avg pChEMBL 8.16
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (535)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZXXCWRYARSIMPM
|
6.5 | Ki | 2 | — | |
ZWURYYOIIRVSAP
|
6.5 | IC50 | 2 | — | |
DRGUVRDBFPDYLQ
|
6.5 | IC50 | 2 | — | |
UNUUFLTUZOLRDF
|
6.5 | IC50 | 2 | — | |
LQXABJNKFHBROP
|
6.5 | IC50 | 2 | — | |
RNNCMVHNZGHSLY
|
6.5 | IC50 | 2 | — | |
AAQHGXPJHYKNDF
|
6.5 | IC50 | 2 | — | |
AAKCZJIYTMOXJF
|
6.5 | IC50 | 2 | — | |
DKRMKDLKTIKQIE
|
6.4 | IC50 | 2 | — | |
RVPUUZJPJXYOSN
|
6.4 | IC50 | 2 | — | |
PTGZJENBFJFKND
|
6.4 | IC50 | 2 | — | |
KSOOVOZETWHNBV
|
6.4 | Ki | 2 | — | |
VRCKDEMDFQJSQX
|
6.4 | IC50 | 2 | — | |
JXZLHWXGEORAOB
|
6.3 | IC50 | 2 | — | |
WOQBGOSNHKHPRH
|
6.3 | IC50 | 2 | — | |
NWZLYDCUPZYBAX
|
6.3 | IC50 | 2 | — | |
XGEPLEYWMXVDFS
|
6.2 | IC50 | 2 | — | |
DIAOYWORMSQRFB
|
6.2 | IC50 | 2 | — | |
JGCMJLQTOLPTCY
|
6.2 | IC50 | 2 | — | |
KRTXDXIJWFIGGJ
|
6.2 | IC50 | 2 | — | |
DYHGVCADLVCJGZ
|
6.2 | IC50 | 2 | — | |
KNFNMFRIDTZZML
|
6.2 | IC50 | 2 | — | |
JGEXEIBPRHWMSL
|
6.1 | IC50 | 2 | — | |
VRQCDTCXZAZNSU
|
6.1 | IC50 | 2 | — | |
HOPRHFCRDCRJAB
|
6.1 | IC50 | 2 | — | |
OTPDSJIKVVZMFC
|
6.1 | IC50 | 2 | — | |
SRYQEUIBRIIYSG
|
6.1 | IC50 | 2 | — | |
IFLIQLQVUMXNFU
|
6.1 | Ki | 2 | — | |
NBEGSXJDADJYHX
|
6.1 | IC50 | 2 | — | |
BXLBQHJYUPJUAV
|
6.0 | IC50 | 2 | — | |
FWTFRDCXSJWXPR
|
6.0 | IC50 | 2 | — | |
GINOPQFPTRYBHX
|
6.0 | IC50 | 2 | — | |
IJWIKFGUGIKEKW
|
6.0 | IC50 | 2 | — | |
SMHWDEHOXGVPME
|
6.0 | IC50 | 2 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — |