Target Details
| UniProt AC | P25101 |
|---|---|
| Gene Symbol | EDNRA |
| Protein Name | Endothelin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 535
- Clinical molecules 0
- Avg pChEMBL 8.16
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (535)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QSPLUDJQEFUAHB
|
7.0 | IC50 | 2 | — | |
TZPUDTSXRNOQNK
|
7.0 | Ki | 2 | — | |
PYYAHQASPOJSMT
|
7.0 | IC50 | 2 | — | |
VKZGOHFGTOOZHY
|
6.9 | IC50 | 2 | — | |
HXUVUUFEMYJLDB
|
6.9 | IC50 | 2 | — | |
CHLXSJALJVYDID
|
6.9 | IC50 | 2 | — | |
HMDVOILXHRHOGL
|
6.9 | IC50 | 2 | — | |
YJMPVDOQESXRRN
|
6.9 | IC50 | 2 | — | |
OZBAKTZMSBVKFA
|
6.9 | IC50 | 2 | — | |
PZBFMEKBVYTVOD
|
6.9 | IC50 | 2 | — | |
RUXNEULYFPIVIB
|
6.9 | IC50 | 2 | — | |
XTHFKSGQJGECGR
|
6.9 | IC50 | 2 | — | |
DTRNHYYWARQBED
|
6.9 | IC50 | 2 | — | |
LQWGCVIETCFLOP
|
6.9 | IC50 | 2 | — | |
ZHGGJHSZAGTHLS
|
6.9 | Ki | 2 | — | |
GQPZSZRJZWLIAV
|
6.9 | IC50 | 2 | — | |
PTWFHEZPRLYXKX
|
6.9 | IC50 | 2 | — | |
YZCIBWHZHRZYCF
|
6.9 | IC50 | 2 | — | |
RQNOIZBVICJIJP
|
6.8 | IC50 | 2 | — | |
ZMUVTNWMWOXWGB
|
6.8 | IC50 | 2 | — | |
QZLAMPMKCJHEKL
|
6.8 | IC50 | 2 | — | |
ZGXRPHUWXAFFDA
|
6.8 | IC50 | 2 | — | |
BWMGPBPXTCNARL
|
6.8 | Ki | 2 | — | |
NXZDWYHCLMUTOJ
|
6.8 | IC50 | 2 | — | |
RLZUSDGCLWDQGG
|
6.8 | IC50 | 2 | — | |
OGGZHZAVIHOULX
|
6.8 | IC50 | 2 | — | |
UUIMPPMXRVSIPX
|
6.8 | IC50 | 2 | — | |
JYYUWMLSDGSJDK
|
6.8 | IC50 | 2 | — | |
USENLZLFWBYRHY
|
6.8 | IC50 | 2 | — | |
WITCSGJQNAEGBT
|
6.8 | IC50 | 2 | — | |
MRISGPUEHMXCRJ
|
6.8 | IC50 | 2 | — | |
BMROGBGRQLVZIB
|
6.8 | IC50 | 2 | — | |
BUZZXSDSIRQVKH
|
6.8 | IC50 | 2 | — | |
WLIQAZXJDQKSEC
|
6.7 | IC50 | 2 | — | |
ZDGQZBNPWPRKMF
|
6.7 | IC50 | 2 | — | |
IBNKZYKCCCSKLB
|
6.7 | IC50 | 2 | — | |
HPSVGPXJVPTNPI
|
6.7 | IC50 | 2 | — | |
UZDORQWMYRRLQV
|
6.7 | IC50 | 2 | — | |
WZQLNTRMQXKHIJ
|
6.7 | Ki | 2 | — | |
XNUQKPOLJGKCNN
|
6.7 | IC50 | 2 | — | |
FVWWHXXCNJDXHS
|
6.7 | IC50 | 2 | — | |
RIFDNBGSPYSLKK
|
6.6 | Ki | 2 | — | |
PGDSQHCYBSJOHQ
|
6.6 | IC50 | 2 | — | |
RDVHLMJRZJBHMF
|
6.6 | Ki | 2 | — | |
VQUBCMKIGJZUME
|
6.6 | Ki | 2 | — | |
DUQYMBAKMGPNBF
|
6.6 | IC50 | 2 | — | |
KWLKTEPEDKFNSG
|
6.6 | IC50 | 2 | — | |
IDXPJQIRPCXAEL
|
6.6 | IC50 | 2 | — | |
YQOHFDDJNGNMBZ
|
6.6 | IC50 | 2 | — | |
IJKPAPFBDVRAPA
|
6.5 | IC50 | 2 | — |