Target Details
| UniProt AC | P25101 |
|---|---|
| Gene Symbol | EDNRA |
| Protein Name | Endothelin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 535
- Clinical molecules 0
- Avg pChEMBL 8.16
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (535)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XCDYCRJUBJSYLD
|
11.4 | Ki | 2 | — | |
AOOKNPITEDSSNB
|
11.3 | Ki | 2 | — | |
XPBBDUYWSIZCNR
|
11.3 | Ki | 2 | — | |
LNPRLVTXUXFAEN
|
11.1 | Ki | 2 | — | |
AXFKGEZDVMCYEO
|
11.0 | Ki | 2 | — | |
CJGRNBWHDOSFES
|
11.0 | Ki | 2 | — | |
CICVRMZHTUTILV
|
11.0 | IC50 | 2 | — | |
HWNXCQQEFQWPHX
|
11.0 | IC50 | 2 | — | |
GJLMSZJTTPBCHM
|
10.8 | IC50 | 2 | — | |
VYAFCUPPLXQIIN
|
10.8 | Ki | 2 | — | |
HKMVKDPUVNFFAO
|
10.7 | Ki | 2 | — | |
XZYQXDCTRBGYKO
|
10.7 | IC50 | 2 | — | |
KYIGOCCCBXRHNJ
|
10.6 | IC50 | 43 | — | |
IDRPGYTWDRQQOE
|
10.6 | IC50 | 2 | — | |
DWNNWTCEZHVDLU
|
10.6 | IC50 | 2 | — | |
IUHMIOAKWHUFKU
|
10.5 | Ki | 2 | — | |
QXJMSZDXBBMLGU
|
10.5 | Ki | 2 | — | |
ZPWXQORYIQFGQB
|
10.5 | IC50 | 2 | — | |
MOTJMGVDPWRKOC
|
10.5 | IC50 | 2 | — | |
JNAFKCJWVUJAQU
|
10.4 | Ki | 2 | — | |
KMOYVJSVLLXFQU
|
10.4 | Ki | 2 | — | |
QGMUOSXKQHPOGD
|
10.4 | Ki | 2 | — | |
XVGVBINHYILTRX
|
10.3 | Ki | 2 | — | |
YQDGZNPRSNHCNL
|
10.3 | IC50 | 2 | — | |
HAZBSXKXEZHGFW
|
10.3 | IC50 | 2 | — | |
FIMDOJGUQJFHTD
|
10.3 | IC50 | 2 | — | |
TWNPZFARHUKPBV
|
10.3 | Ki | 2 | — | |
XPPNYNZMOQSBAA
|
10.3 | Ki | 2 | — | |
WERWDDKHJRXHAF
|
10.2 | IC50 | 2 | — | |
KBHRSNOQJNLUNL
|
10.2 | IC50 | 2 | — | |
FVNKNOUQLKAPJI
|
10.2 | IC50 | 2 | — | |
YAWKZANKTNYRSZ
|
10.2 | IC50 | 2 | — | |
JVWVTPZZEHLARL
|
10.1 | IC50 | 2 | — | |
MOTJMGVDPWRKOC
|
10.1 | IC50 | 2 | — | |
KNCYVPWSDRUANJ
|
10.1 | IC50 | 2 | — | |
LDYLIYKANSSERK
|
10.0 | IC50 | 2 | — | |
WQULYHKGCLHTBZ
|
10.0 | IC50 | 2 | — | |
WELUHUKTVXHVBY
|
10.0 | IC50 | 2 | — | |
GYPOJYXMDPSAQP
|
10.0 | IC50 | 2 | — | |
KJNNBRVUQZDOET
|
10.0 | Ki | 2 | — | |
MIDBNMYTUQUADA
|
9.9 | Ki | 2 | — | |
NRCLKFNYCQXXAL
|
9.9 | IC50 | 2 | — | |
YGGFLIPTDYLEIC
|
9.9 | IC50 | 2 | — | |
MCHCGWZNXSZKJY
|
9.9 | Ki | 2 | — | |
SISHUQWGICPIJE
|
9.9 | IC50 | 2 | — | |
VHHUBYWYNJXLPT
|
9.8 | Ki | 2 | — | |
ZUBDGKVDJUIMQQ
|
9.8 | IC50 | 2 | — | |
JPPYWKVKLSBQJM
|
9.7 | Ki | 2 | — | |
GAZYTXSFOKMUAC
|
9.7 | IC50 | 2 | — | |
IECXSVOMLVKXGN
|
9.7 | IC50 | 2 | — |