Target Details
| UniProt AC | P25098 |
|---|---|
| Gene Symbol | GRK2 |
| Protein Name | Beta-adrenergic receptor kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00169 (PH) PF00069 (Pkinase) PF00615 (RGS) |
Summary
- Multi-target molecules 141
- Clinical molecules 1
- Avg pChEMBL 7.33
KEGG Pathways (6)
Active Molecules (141)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CDRCHNJBVCLMFS
|
6.9 | IC50 | 2 | — | |
QFADBQQWVFQUHB
|
6.9 | IC50 | 2 | — | |
GMDDIUVOWBJMQH
|
6.8 | IC50 | 2 | — | |
SGGQLVSCPDXQCB
|
6.8 | IC50 | 2 | — | |
BLMBNKDQXGINRE
|
6.8 | IC50 | 3 | — | |
COZSHMVZWUUCPG
|
6.8 | IC50 | 2 | — | |
DXXLHEZKXIIHMT
|
6.8 | IC50 | 2 | — | |
LYADGAGFYYXXIO
|
6.8 | IC50 | 82 | — | |
XBRPSBXARPNOBH
|
6.8 | IC50 | 2 | — | |
IIRWNGPLJQXWFJ
|
6.8 | Kd | 21 | — | |
BXTYCBBDHNQJNG
|
6.7 | IC50 | 3 | — | |
SCUPKXISFBICSC
|
6.7 | IC50 | 2 | — | |
QTCMCOOGSCOKGD
|
6.6 | IC50 | 2 | — | |
VHISWSDHEWXRKH
|
6.6 | IC50 | 2 | — | |
SRDLWBLWLYRNNX
|
6.6 | IC50 | 2 | — | |
IGPLDYDCTCCRIM
|
6.5 | IC50 | 2 | — | |
UGYAZGXSMRGKRD
|
6.5 | IC50 | 3 | — | |
PQEUUIPIJGRXTL
|
6.5 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
6.4 | Kd | 1075 | — | |
BSBBIWMXRBLRGQ
|
6.4 | IC50 | 2 | — | |
JPDACOLMZSWYPX
|
6.3 | IC50 | 2 | — | |
AGVLCYIXOACYIT
|
6.3 | IC50 | 2 | — | |
MWVKLRSIDOXBSE
|
6.3 | IC50 | 4 | — | |
VGSYMGCEDYSPMI
|
6.3 | IC50 | 2 | — | |
JYIQDDWOZUMLLE
|
6.3 | IC50 | 2 | — | |
WRBFHBIIEVVYIJ
|
6.3 | IC50 | 2 | — | |
QCLXNOBXQUWUEW
|
6.3 | IC50 | 9 | — | |
QNABDSWBQJKBHK
|
6.2 | IC50 | 45 | — | |
XWCWGOOBIPAWPA
|
6.2 | IC50 | 2 | — | |
CWUZHXXAZSEESR
|
6.2 | IC50 | 3 | — | |
JNVSJVSIHCPPTE
|
6.2 | IC50 | 2 | — | |
HEAIGWIZTYAQTC
|
6.1 | IC50 | 2 | — | |
POEIXYXZODKFHQ
|
6.1 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
6.1 | IC50 | 408 | — | |
XMPOFQWNHXAUKI
|
6.0 | IC50 | 2 | — | |
UDRONCPPXHIFAY
|
6.0 | IC50 | 2 | — | |
BBDOLYGGPDFTSD
|
6.0 | Ki | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
SGPKBJQYKUQGKV
|
6.0 | Ki | 3 | — |