Target Details
| UniProt AC | P25098 |
|---|---|
| Gene Symbol | GRK2 |
| Protein Name | Beta-adrenergic receptor kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00169 (PH) PF00069 (Pkinase) PF00615 (RGS) |
Summary
- Multi-target molecules 141
- Clinical molecules 1
- Avg pChEMBL 7.33
KEGG Pathways (6)
Active Molecules (141)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PNLQOSABVUZYHX
|
7.8 | IC50 | 2 | — | |
CYINSAOYPJZRPS
|
7.7 | IC50 | 2 | — | |
RAFDCMBISGTRKN
|
7.7 | IC50 | 2 | — | |
JOJIACUBCDTHHJ
|
7.7 | IC50 | 2 | — | |
VWBSMGFTNCQOMB
|
7.7 | IC50 | 3 | — | |
BBZVXUBFCDUWHJ
|
7.7 | IC50 | 2 | — | |
QCDDREXJCIDOSP
|
7.6 | IC50 | 2 | — | |
OTNWPJUPTWXBRM
|
7.6 | IC50 | 2 | — | |
WFOVEDJTASPCIR
|
7.5 | IC50 | 2 | — | |
FJHLPXVADZHKER
|
7.5 | IC50 | 2 | — | |
YUSNFTGATCSSBA
|
7.4 | IC50 | 2 | — | |
FENQBUSSSWWVGH
|
7.4 | IC50 | 3 | — | |
VZALQQCVHAISSG
|
7.4 | IC50 | 2 | — | |
LNHMXIAOIPMUFG
|
7.4 | IC50 | 2 | — | |
AHHBKDVMDHSKFS
|
7.4 | IC50 | 2 | — | |
XYUFCXJZFZPEJD
|
7.4 | IC50 | 23 | Yes | |
LESAWXMGKBXNAN
|
7.4 | IC50 | 2 | — | |
ACHYMSFHZAUMEM
|
7.3 | IC50 | 2 | — | |
RLCLKOKLWUPURE
|
7.3 | IC50 | 2 | — | |
ZKFHBBAGQQHMMG
|
7.3 | IC50 | 2 | — | |
LHAZDFBNDIQNSG
|
7.3 | IC50 | 4 | — | |
ZHDPMPLGMKQADI
|
7.3 | IC50 | 3 | — | |
ASPDMKGCEMLVBM
|
7.2 | IC50 | 2 | — | |
IETGNPWDJMSKGZ
|
7.2 | IC50 | 2 | — | |
MSYSXAOSMCNJKL
|
7.2 | IC50 | 3 | — | |
SVKLMBZNMVZHTI
|
7.2 | IC50 | 2 | — | |
BXMIHYGPXLIJBT
|
7.0 | Ki | 2 | — | |
DCJIPWKGABWYAG
|
7.0 | Ki | 2 | — | |
GKLCWXCSSBEZOG
|
7.0 | Ki | 2 | — | |
HDOAZITZHWAPBC
|
7.0 | Ki | 2 | — | |
HTBWNFFLHDWPKO
|
7.0 | Ki | 2 | — | |
KWGIZLMNJXFPFV
|
7.0 | Ki | 3 | — | |
KYWXYKMZNMJBMK
|
7.0 | Ki | 2 | — | |
KZZVYUYRNIMTBP
|
7.0 | IC50 | 2 | — | |
NDSSSMYGJDDEPB
|
7.0 | Ki | 3 | — | |
PDXVRCZNPFLZJP
|
7.0 | Ki | 3 | — | |
PWMGIYOLYSEHBN
|
7.0 | Ki | 3 | — | |
QDNSHFHBLOTJEL
|
7.0 | Ki | 3 | — | |
QNWKTVKWUCLLKW
|
7.0 | Ki | 2 | — | |
RPBKUXXUYPWIPS
|
7.0 | Ki | 3 | — | |
VFKYFTQIVJAIAA
|
7.0 | Ki | 2 | — | |
VRKITNLDCQGIJI
|
7.0 | Ki | 3 | — | |
XHFJYOGNWBJZAX
|
7.0 | Ki | 2 | — | |
XMRRJWMAVDAELT
|
7.0 | Ki | 2 | — | |
YKAVZWRGBOWKDP
|
7.0 | IC50 | 2 | — | |
YKLNVZIGQDKBKJ
|
7.0 | Ki | 3 | — | |
ZXYUSNLUAQYJFK
|
7.0 | Ki | 3 | — | |
RAXZSEGXMBWYQK
|
7.0 | Kd | 21 | — | |
YJQKIQOVJOGHMP
|
6.9 | IC50 | 2 | — | |
ANLHPWBHGQANDX
|
6.9 | IC50 | 2 | — |