Target Details
| UniProt AC | P25098 |
|---|---|
| Gene Symbol | GRK2 |
| Protein Name | Beta-adrenergic receptor kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00169 (PH) PF00069 (Pkinase) PF00615 (RGS) |
Summary
- Multi-target molecules 141
- Clinical molecules 1
- Avg pChEMBL 7.33
KEGG Pathways (6)
Active Molecules (141)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IXXFFNLFAIHVPM
|
8.8 | IC50 | 2 | — | |
DMNINFHJFPFPIZ
|
8.7 | IC50 | 4 | — | |
NVEGMPXYWCBLOA
|
8.7 | IC50 | 2 | — | |
MLCHXEPEMWHPKH
|
8.7 | IC50 | 7 | — | |
UCVRLTXXBKZAOV
|
8.6 | IC50 | 5 | — | |
QHMDGFUUSLLYGF
|
8.5 | IC50 | 2 | — | |
ADUQCZZLBHMOBQ
|
8.5 | IC50 | 4 | — | |
ITHPWIHYZQLUIG
|
8.5 | IC50 | 7 | — | |
YBLPMNNVXVEMKC
|
8.4 | IC50 | 5 | — | |
AJPNQVZYWOGOKN
|
8.4 | IC50 | 5 | — | |
APIVUJRBRZKGIM
|
8.4 | IC50 | 2 | — | |
ZODPLLYTMWNTCA
|
8.4 | IC50 | 7 | — | |
FJXAKWGPTCSFIG
|
8.4 | IC50 | 7 | — | |
QZCITBQFXYREEJ
|
8.3 | IC50 | 7 | — | |
LTDFDPHSEHTUCI
|
8.3 | IC50 | 5 | — | |
AEAIPRJCBYGHJK
|
8.3 | IC50 | 2 | — | |
QQJKCGXOHWHBQV
|
8.2 | IC50 | 4 | — | |
XWJOKKXDMHSILW
|
8.2 | IC50 | 3 | — | |
YIAIWVFWUCOYKA
|
8.2 | IC50 | 4 | — | |
XQKRWDLELRIZOC
|
8.2 | IC50 | 7 | — | |
SGOFJRIGAKFXAH
|
8.2 | IC50 | 6 | — | |
ARSZMAAOVNYKQN
|
8.1 | IC50 | 3 | — | |
FVEIPMUKOTZXBA
|
8.1 | IC50 | 7 | — | |
DFYJVEZNHJSNLL
|
8.1 | IC50 | 2 | — | |
PXKQKKHBHPRTEG
|
8.1 | IC50 | 6 | — | |
RAOPEUTYHRNFHJ
|
8.1 | IC50 | 7 | — | |
ULMMSSXMAQOVME
|
8.1 | IC50 | 7 | — | |
YWKCCOXVWMNFSF
|
8.1 | IC50 | 7 | — | |
OVBAFUGPHNUQFH
|
8.1 | IC50 | 7 | — | |
XNLQUWXXCRJCDC
|
8.1 | IC50 | 4 | — | |
BDLBLCWMNJLLLI
|
8.1 | IC50 | 5 | — | |
ICVWYIZCPUIPOY
|
8.1 | IC50 | 7 | — | |
FNAWEKRTBLXUJI
|
8.1 | IC50 | 7 | — | |
QTMWJQCPEOTFSB
|
8.1 | IC50 | 5 | — | |
UWZBUGMYQWUJLU
|
8.1 | IC50 | 5 | — | |
WOBKYDKXSVLQGJ
|
8.1 | IC50 | 7 | — | |
FMUUGBFOPCVEBP
|
8.0 | IC50 | 7 | — | |
PUELPOFWJXDUSU
|
8.0 | IC50 | 4 | — | |
ZLPVQTFOPHTMQK
|
8.0 | IC50 | 4 | — | |
SKZTUPIPRLPDKY
|
8.0 | Ki | 3 | — | |
UQHPGIWKYQJUIE
|
8.0 | IC50 | 7 | — | |
WGESQHUBLPGDDK
|
8.0 | IC50 | 3 | — | |
HMUYSTSHIXJVRO
|
8.0 | IC50 | 5 | — | |
GEPQSMPOMLNHIV
|
7.9 | IC50 | 2 | — | |
QVDUXSXBOMFTNR
|
7.9 | IC50 | 3 | — | |
XKLOPDYWVXDVPR
|
7.9 | IC50 | 2 | — | |
LKHWQSZVOZRQIZ
|
7.9 | IC50 | 6 | — | |
NKZKSFKCRMCQQH
|
7.8 | IC50 | 2 | — | |
ZEZFDAXYOWUZPP
|
7.8 | IC50 | 2 | — | |
VPSTUMWWEPHXGY
|
7.8 | IC50 | 2 | — |