Target Details
| UniProt AC | P25084 |
|---|---|
| Gene Symbol | lasR |
| Protein Name | Transcriptional activator protein LasR |
| Organism | Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22644 / CIP 104116 / JCM 14847 / LMG 12228 / 1C / PRS 101 / PAO1) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF03472 (Autoind_bind) PF00196 (GerE) |
Summary
- Multi-target molecules 4
- Clinical molecules 0
- Avg pChEMBL 6.65
Active Molecules (4)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XXSUYIPTSOFKRD
|
7.5 | IC50 | 2 | — | |
TZWZKDULKILUPV
|
6.6 | IC50 | 2 | — | |
JKEJEOJPJVRHMQ
|
6.5 | IC50 | 2 | — | |
ZYWNMRPOYLXAAW
|
6.0 | IC50 | 2 | — |