Target Details
| UniProt AC | P25025 |
|---|---|
| Gene Symbol | CXCR2 |
| Protein Name | C-X-C chemokine receptor type 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 224
- Clinical molecules 0
- Avg pChEMBL 7.63
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (224)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JVOHPOBSHINFNU
|
6.4 | IC50 | 2 | — | |
ZKLITWMNDRXOLR
|
6.4 | Ki | 2 | — | |
PSPSMPJFVZTXSD
|
6.4 | Ki | 2 | — | |
TVANIYMHXPLFFL
|
6.4 | IC50 | 2 | — | |
HKRNYOZJJMFDBV
|
6.4 | IC50 | 2 | — | |
VOAPNZIKRKHEHR
|
6.4 | IC50 | 2 | — | |
QORPNJQYKGLIAV
|
6.3 | Ki | 2 | — | |
UDGYWARCEKJDIJ
|
6.3 | Ki | 2 | — | |
LYZBESBXJHUNLT
|
6.3 | Ki | 2 | — | |
XCVNKDBFHMYYDO
|
6.3 | Ki | 2 | — | |
XHLNLGDWWRFFBW
|
6.3 | Ki | 2 | — | |
BAWCTQVXGNPSAG
|
6.2 | Ki | 2 | — | |
KJEUTTLHSRWQMD
|
6.2 | Ki | 2 | — | |
YIKGYASPCLWXCD
|
6.2 | Ki | 2 | — | |
UKBAGMZMGJKUER
|
6.2 | IC50 | 2 | — | |
KCIRBTXGALUYHT
|
6.2 | IC50 | 2 | — | |
QMQGUUOGRMUXFL
|
6.2 | IC50 | 2 | — | |
DGGJPUBUCAEEHT
|
6.1 | IC50 | 2 | — | |
MWABJGSIPHBDDC
|
6.1 | Ki | 2 | — | |
AHAOUMFJVVZFDM
|
6.1 | IC50 | 2 | — | |
UUNDOBHSENXEFU
|
6.0 | IC50 | 2 | — | |
COQNFUICOUPODA
|
6.0 | Ki | 2 | — | |
OISJPBYRKOJZRI
|
6.0 | IC50 | 2 | — | |
PFVOSGMAMDBGFG
|
6.0 | IC50 | 2 | — |