Target Details
| UniProt AC | P25025 |
|---|---|
| Gene Symbol | CXCR2 |
| Protein Name | C-X-C chemokine receptor type 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 224
- Clinical molecules 0
- Avg pChEMBL 7.63
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (224)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PPCFLIBERCNFID
|
7.2 | IC50 | 2 | — | |
SIUQYAWDXLUCLD
|
7.2 | IC50 | 2 | — | |
TXIZIPIJZWQRPG
|
7.2 | Ki | 2 | — | |
DGPHJNJINCRCKW
|
7.2 | IC50 | 5 | — | |
HCGUUQDQSYMJAU
|
7.2 | IC50 | 2 | — | |
BIVKRDOOTZFPRA
|
7.2 | IC50 | 2 | — | |
KBLOFZHBIDLNIS
|
7.1 | IC50 | 2 | — | |
MMVFNAGMKWQAKS
|
7.1 | IC50 | 4 | — | |
QUKXEAVCHJVKEA
|
7.1 | IC50 | 2 | — | |
GMNNTQPTKYJUKQ
|
7.1 | IC50 | 2 | — | |
IJPNBRULEFKYSA
|
7.1 | Ki | 2 | — | |
KQDRVXQXKZXMHP
|
7.1 | IC50 | 2 | — | |
LOSWDIGGZMWFHV
|
7.1 | Ki | 2 | — | |
WYWJXUDCXPYMIQ
|
7.1 | Ki | 2 | — | |
MXDWNZUMSIYAFL
|
7.1 | IC50 | 2 | — | |
LQUGDEWJKLEGOJ
|
7.1 | IC50 | 2 | — | |
PCXDKTNTSYUMHN
|
7.1 | IC50 | 2 | — | |
XEJUWHPWBDYKSK
|
7.1 | IC50 | 2 | — | |
VWSXKWXISJLOQM
|
7.0 | IC50 | 6 | — | |
APDVPDFSMORZLD
|
7.0 | IC50 | 2 | — | |
HEFNNWSXXWATRW
|
7.0 | IC50 | 5 | — | |
SAJPPXKBUXNTKQ
|
7.0 | Ki | 2 | — | |
SJWVRSVJDTUULR
|
7.0 | IC50 | 2 | — | |
HEFNNWSXXWATRW
|
7.0 | IC50 | 3 | — | |
JBBKREGWJICILL
|
7.0 | IC50 | 2 | — | |
QIBUUCFTHGXSFM
|
7.0 | IC50 | 2 | — | |
SGLBQNTUAMMYTP
|
7.0 | IC50 | 2 | — | |
KBLOFZHBIDLNIS
|
6.9 | IC50 | 2 | — | |
LUNAFTMLJLEOEQ
|
6.9 | Ki | 2 | — | |
NPKHWEBWIFDKHH
|
6.9 | IC50 | 2 | — | |
MUMCBMXUGZFFMH
|
6.8 | Ki | 2 | — | |
WCBDQNUHQNEQLF
|
6.8 | IC50 | 2 | — | |
YRQLRCRBEYSAIN
|
6.8 | IC50 | 4 | — | |
UXUIKTKXWYNOMQ
|
6.8 | Ki | 2 | — | |
ASWBTVXNCFSFOM
|
6.8 | IC50 | 2 | — | |
FVQFHIDXFRDHQK
|
6.7 | Ki | 2 | — | |
KCVWGCOBGFLUEB
|
6.7 | IC50 | 5 | — | |
OISJPBYRKOJZRI
|
6.7 | IC50 | 2 | — | |
VZNLCSKTOPAQML
|
6.7 | IC50 | 2 | — | |
IAGWEZFSRRPOSS
|
6.7 | Ki | 2 | — | |
HVAOCXFQAGCNQP
|
6.7 | Ki | 2 | — | |
OISJPBYRKOJZRI
|
6.7 | IC50 | 2 | — | |
WKNNSCHBIPUNFV
|
6.7 | Ki | 2 | — | |
YFTUGOHVHFFSHQ
|
6.7 | IC50 | 2 | — | |
ZMLPGOTZQCYELQ
|
6.7 | IC50 | 2 | — | |
MXCRXBCGEWUMNZ
|
6.5 | IC50 | 2 | — | |
DXPCTOZNUCZJPC
|
6.5 | Ki | 2 | — | |
FIBJPCXODZVPBQ
|
6.5 | Ki | 2 | — | |
BKQNUKCQBYWSPK
|
6.5 | Ki | 2 | — | |
STUJFSIJLYQOCY
|
6.4 | IC50 | 2 | — |