Target Details
| UniProt AC | P25025 |
|---|---|
| Gene Symbol | CXCR2 |
| Protein Name | C-X-C chemokine receptor type 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 224
- Clinical molecules 0
- Avg pChEMBL 7.63
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (224)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GULGFHPSYNQMBP
|
7.9 | IC50 | 2 | — | |
NEZMHIVTYRWBEX
|
7.9 | IC50 | 2 | — | |
OQCIAVOJSLDHHC
|
7.9 | Ki | 2 | — | |
IYZWLQHDOCJREA
|
7.9 | IC50 | 2 | — | |
WWSNTFDUUVNWIC
|
7.9 | Ki | 2 | — | |
IPLGVPPLWIAZSG
|
7.8 | Ki | 2 | — | |
NICQNGMZJXZBJM
|
7.8 | Ki | 2 | — | |
KBLOFZHBIDLNIS
|
7.8 | IC50 | 5 | — | |
NTWHZYBSKKHULS
|
7.8 | IC50 | 2 | — | |
RZXVFVRPSNXVEC
|
7.8 | IC50 | 2 | — | |
CODGMHXCDXLYFF
|
7.8 | IC50 | 2 | — | |
SSBIYBNARHHMGE
|
7.8 | Ki | 2 | — | |
UTDWJMBRBOKFJV
|
7.8 | IC50 | 2 | — | |
CBIODTKCFBGXHU
|
7.8 | IC50 | 2 | — | |
SPLGZZDGUQTEHE
|
7.8 | IC50 | 5 | — | |
XZVGETAASKRSBI
|
7.7 | Ki | 2 | — | |
BGHMYZUFTBKLKU
|
7.7 | IC50 | 2 | — | |
JBBKREGWJICILL
|
7.7 | IC50 | 5 | — | |
KRRJDGLUFFFYHX
|
7.7 | IC50 | 2 | — | |
VNUFOKWSYSXHCN
|
7.7 | Ki | 2 | — | |
QEOSQTDOWDCAEV
|
7.7 | Kd | 2 | — | |
AEDMWJARWOMJKQ
|
7.7 | IC50 | 2 | — | |
MSJKBTMMJKJYHB
|
7.7 | IC50 | 2 | — | |
XETXTFIIXKTWPQ
|
7.6 | IC50 | 2 | — | |
MCQSWTLKUIEWQM
|
7.6 | Ki | 2 | — | |
ZHAAHVPYFDDLLE
|
7.6 | IC50 | 2 | — | |
MRHPZVNAGXMSIH
|
7.6 | IC50 | 2 | — | |
BGXSRDRXCPKCLB
|
7.5 | IC50 | 2 | — | |
HDQNDRCZSVEGSG
|
7.5 | IC50 | 5 | — | |
MQBZVUNNWUIPMK
|
7.5 | IC50 | 3 | — | |
XBPBJDFJAWKYCK
|
7.5 | IC50 | 2 | — | |
ZHOSAEFOHKXJDJ
|
7.5 | IC50 | 5 | — | |
YWEPAFKNLSBBBU
|
7.5 | IC50 | 3 | — | |
DKYWVDODHFEZIM
|
7.5 | IC50 | 3 | — | |
UNPQYPMTWSIZRR
|
7.4 | IC50 | 2 | — | |
HDQNDRCZSVEGSG
|
7.4 | IC50 | 2 | — | |
SIUQYAWDXLUCLD
|
7.4 | IC50 | 4 | — | |
VZRIHFZJVIOJBE
|
7.4 | IC50 | 2 | — | |
CMANXHXTSWTYRG
|
7.4 | IC50 | 2 | — | |
SHLGVUBRPWNMLF
|
7.4 | IC50 | 2 | — | |
FNGBYTBDUQDISM
|
7.4 | IC50 | 2 | — | |
LPLKAXWKZWWASO
|
7.4 | IC50 | 2 | — | |
QPFHUUXBBCZCOF
|
7.4 | IC50 | 2 | — | |
SCSNKXZAGMCAGA
|
7.4 | Ki | 2 | — | |
WOBYQWNRYZGWRU
|
7.4 | IC50 | 2 | — | |
YTTGJPIBJUDFQG
|
7.3 | IC50 | 2 | — | |
MNULHNJDCIVGAO
|
7.3 | Kd | 2 | — | |
DKYWVDODHFEZIM
|
7.3 | IC50 | 4 | — | |
KMOKWTXCNPBSHR
|
7.3 | IC50 | 2 | — | |
DLHXKIOUORFOQU
|
7.3 | IC50 | 2 | — |